Publication: Heterospirocyclic 3-Amino-2H-azirines as Convenient Building Blocks in Peptide Synthesis
Heterospirocyclic 3-Amino-2H-azirines as Convenient Building Blocks in Peptide Synthesis
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Strässler, C., & Heimgartner, H. (2019). Heterospirocyclic 3-Amino-2H-azirines as Convenient Building Blocks in Peptide Synthesis. Heterocycles, 99(1), 446. https://doi.org/10.3987/COM-18-S(F)41
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Heterospirocyclic 3-amino-2H-azirines with a tetrahydropyran (Thp), tetrahydrothiopyran (Tht), or N-protected piperidine (Pip) moiety are useful reagents for the preparation of peptides containing the corresponding six-membered heterocyclic 4-amino-4-carboxylic acid unit. In the present study, tripeptides of the type H-Asp-D-Ala-Xaa-OMe, where Xaa is the heterocyclic amino acid, were prepared according to the ‘azirine/oxazolone method’.
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- Strässler, Christoph
- Heimgartner, Heinz
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Strässler, C., & Heimgartner, H. (2019). Heterospirocyclic 3-Amino-2H-azirines as Convenient Building Blocks in Peptide Synthesis. Heterocycles, 99(1), 446. https://doi.org/10.3987/COM-18-S(F)41
