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Nievergelt, Philipp; Berliat, Florian; McAuley, Katherine E; Dorgan, Colin R; van Well, Renate Maria; Thorn, Andrea; Spingler, Bernhard (2024). RNA oligomers at atomic resolution containing 1‐methylpseudouridine, an essential building block of mRNA vaccines. ChemMedChem, 19(7):e202300600.

Braschler, Lorin; Thuany, Mabliny; de Lira, Claudio A B; Scheer, Volker; Nikolaidis, Pantelis T; Weiss, Katja; Knechtle, Beat (2024). Personality of marathon runners: a narrative review of recent findings. EXCLI Journal, 23:441-474.

Brugger, Daniel; Wilhelm, Belinda; Schusser, Benjamin; Gisch, Nicolas; Matthes, Julia; Zhao, Jie; Windisch, Wilhelm (2024). Masson Pine pollen (Pinus massoniana) activate HD11 chicken macrophages in vitro. Journal of Ethnopharmacology, 325:117870.

Csucker, Joshua; Decrausaz, Nathalie; Jäggi, Sarah Isabella; Blacque, Olivier; Spingler, Bernhard; Alberto, Roger (2024). Synthesis and Photophysical Evaluation of 3,3’‐Nitrogen Bis‐Substituted <i>fac</i>‐[Re(CO)<sub>3</sub>(Diimine)Br] Complexes. Helvetica Chimica Acta, 107(2):e202300239.


Schreck, Moritz-Valentin; Burgard, Caroline; Schmidtke, Alexander; Hierlmeier, Ina; Stemler, Tobias; Maus, Stephan; Rosar, Florian; Jung, Martin; Speicher, Andreas; Ezziddin, Samer; Holland, Jason P; Bartholomä, Mark D (2023). Radiometal Complexes as Pharmacokinetic Modifiers: A Potent $^{68}$Ga-Labeled Gastrin-Releasing Peptide Receptor Antagonist Based on the Macrocyclic Metal Chelator NODIA-Me. Molecular Pharmaceutics, 20(12):6463-6473.

Vackova, Zuzana; Levenfus, Ian; Pohl, Daniel (2023). Interventional functional diagnostics in gastrointestinal endoscopy: Combining diagnostic and therapeutic tools in the endoscopy suite with the functional lumen imaging probe. Current Opinion in Pharmacology, 73:102414.

Shamarina, Dasha; Sluga-O'Callaghan, Martina; Kassianos, George; Marijam, Alen; Dave, Vaidehi; Davenport, Eric; Andani, Anar; Curran, Desmond; Dewda, Pavitra; Steffen, Robert (2023). Knowledge, Attitudes, and Practices of European Healthcare Professionals towards Hepatitis A and Hepatitis B Vaccination in at-Risk Adults. Vaccines, 11(11):1645.

Hartmann, K Patricia; van Gogh, Merel; Freitag, Patrick C; Kast, Florian; Nagy-Davidescu, Gabriela; Borsig, Lubor; Plückthun, Andreas (2023). FAP-retargeted Ad5 enables in vivo gene delivery to stromal cells in the tumor microenvironment. Molecular Therapy, 31(10):2914-2928.

Schweckendiek, Daniel; Pohl, D (2023). Pharmacologic treatment of gastroparesis: What is (still) on the horizon? Current Opinion in Pharmacology, 72:102395.

Martinez-Navajas, Gonzalo; Ceron-Hernandez, Jorge; Simon, Iris; Lupiañez, Pablo; Diaz-McLynn, Sofia; Perales, Sonia; Modlich, Ute; Guerrero, Jose A; Martin, Francisco; Sevivas, Teresa; Lozano, Maria L; Rivera, Jose; Ramos-Mejia, Veronica; Tersteeg, Claudia; Real, Pedro J (2023). Lentiviral gene therapy reverts GPIX expression and phenotype in Bernard-Soulier syndrome type C. Molecular Therapy : Nucleic Acids, 33:75-92.

Kolkhir, Pavel; Akdis, Cezmi A; Akdis, Mubeccel; Bachert, Claus; Bieber, Thomas; Canonica, Giorgio Walter; Guttman-Yassky, Emma; Metz, Martin; Mullol, Joaquim; Palomares, Oscar; Renz, Harald; Ständer, Sonja; Zuberbier, Torsten; Maurer, Marcus (2023). Type 2 chronic inflammatory diseases: targets, therapies and unmet needs. Nature Reviews. Drug Discovery, 22(9):743-767.

Duminis, Tomas; Heljak, Marcin; Święszkowski, Wojciech; Ereskovsky, Alexander; Dziedzic, Izabela; Nowicki, Marek; Pajewska-Szmyt, Martyna; Voronkina, Alona; Bornstein, Stefan R; Ehrlich, Hermann (2023). On the Mechanical Properties of Microfibre-Based 3D Chitinous Scaffolds from Selected Verongiida Sponges. Marine Drugs, 21(9):463.

Gergely, Lea P; Yüceel, Çiğdem; İşci, Ümit; Spadin, Florentin S; Schneider, Lukas; Spingler, Bernhard; Frenz, Martin; Dumoulin, Fabienne; Vermathen, Martina (2023). Comparing PVP and Polymeric Micellar Formulations of a PEGylated Photosensitizing Phthalocyanine by NMR and Optical Techniques. Molecular Pharmaceutics, 20(8):4165-4183.

Kraehenbuehl, Lukas; Schneider, Stephanie; Pawlik, Laura; Mangana, Joanna; Cheng, Phil; Dummer, Reinhard; Meier-Schiesser, Barbara (2023). Cutaneous Adverse Events of Systemic Melanoma Treatments: A Retrospective Single-Center Analysis. Pharmaceuticals, 16(7):935.

Nikolaidis, Pantelis T; Knechtle, Beat (2023). Predictors of half-marathon performance in male recreational athletes. EXCLI Journal, 22:559-566.

Stoffel, Sandro Tiziano; Schwenkglenks, Matthias; Mutschler, Thomas (2023). General Practitioners' Awareness and Perception of Current Pneumococcal Vaccination for Adult Patients with Known Risk Factors in Switzerland: Evidence from a Survey. Vaccines, 11(6):1101.

Bedi, Rajiv Kumar; Huang, Danzhi; Li, Yaozong; Caflisch, Amedeo (2023). Structure-Based Design of Inhibitors of the m$^{6}$A-RNA Writer Enzyme METTL3. ACS Bio & Med Chem Au, 3(4):359-370.

Auberson, Yves P; Benfatti, Fides; Gillingham, Dennis; Hartrampf, Nina (2023). An Active Member of the EFMC: The Division of Medicinal Chemistry and Chemical Biology of the Swiss Chemical Society. ChemMedChem, 18(11):e202300014.

Oi, Kathryn K; Moehle, Kerstin; Schuster, Matthias; Zerbe, Oliver (2023). Early molecular insights into thanatin analogues binding to A. baumannii LptA. Molecules, 28(11):4335.

Hoff, Lukas V; Schnell, Simon D; Benchimol, Elie; Foutinho, Fabio Pereira; Tomio, Andrea; Rickhaus, Michel; Gademann, Karl (2023). Preparation of 3-Bromo-1,2,4,5-tetrazine. Helvetica Chimica Acta, 106(4):e202200198.

Mohamad-Ramshan, Rukshana; Ande, Chennaiah; Matsushita, Takahiko; Haldimann, Klara; Vasella, Andrea; Hobbie, Sven N; Crich, David (2023). Synthesis of 4-O-(4-Amino-4-deoxy-β-D-xylopyranosyl)paromomycin and 4-S-(β-D-Xylopyranosyl)-4-deoxy-4'-thio-paromomycin and Evaluation of their Antiribosomal and Antibacterial Activity. Tetrahedron, 135:133330.

Morais, Marcos José; de Oliveira, Vinnycius Nunes; Viana, Ricardo Borges; Andrade, Marilia Santos; Vancini, Rodrigo Luiz; Arida, Ricardo Mario; Costa, Gustavo De Conti Teixeira; Campos, Mário Hebling; Vieira, Carlos Alexandre; Weiss, Katja; Knechtle, Beat; de Lira, Claudio Andre Barbosa (2023). Acute effects of moderate-intensity continuous physical exercise performed with different amounts of muscle mass on executive function in healthy young adults: a randomized trial. EXCLI Journal, 22:1032-1046.

Weiss, Katja; Seffrin, Aldo; Andrade, Marilia Santos; Ahmad, Wais; Forte, Pedro; Moreitz, Sascha; Stanula, Arkadiusz; Cuk, Ivan; Nikolaidis, Pantelis Theo; Knechtle, Beat (2023). Where are the fastest master butterfly swimmers competing in the FINA World Masters Championships from? EXCLI Journal, 22:604-619.


Weber, Ronja; Kaeslin, Jérôme; Moeller, Sophia; Perkins, Nathan; Micic, Srdjan; Moeller, Alexander (2022). Effects of a Volatile Organic Compound Filter on Breath Profiles Measured by Secondary Electrospray High-Resolution Mass Spectrometry. Molecules, 28(1):45.

Irziqat, Bahaaeddin; Berger, Jan; Cebrat, Aleksandra; Mendieta‐Moreno, Jesús I; Sundar, Mothuku Shyam; Bedekar, Ashutosh V; Ernst, Karl‐Heinz (2022). Conglomerate Aggregation of 7,12,17-Trioxa[11]helicene into Homochiral Two-Dimensional Crystals on the Cu(100) Surface. Helvetica Chimica Acta, 105(12):e202200114.

Jönsson, Åsa Lina M; Hernando, Nati; Knöpfel, Thomas; Mogensen, Susie; Bendstrup, Elisabeth; Hilberg, Ole; Christensen, Jane Hvarregaard; Simonsen, Ulf; Wagner, Carsten A (2022). Impaired phosphate transport in SLC34A2 variants in patients with pulmonary alveolar microlithiasis. Human Genomics, 16(1):13.

Al-Wahaibi, Lamya H; Alagappan, Kowsalya; Blacque, Olivier; Mohamed, Ahmed A B; Hassan, Hanan M; Percino, María Judith; El-Emam, Ali A; Thamotharan, Subbiah (2022). X-ray Structures and Computational Studies of Two Bioactive 2-(Adamantane-1-carbonyl)-N-substituted Hydrazine-1-carbothioamides. Molecules, 27(23):8425-8443.

Mathes, Sebastian; Fahrner, Alexandra; Luca, Edlira; Krützfeldt, Jan (2022). Growth hormone/IGF-I-dependent signaling restores decreased expression of the myokine SPARC in aged skeletal muscle. Journal of Molecular Medicine, 100(11):1647-1658.

Al-Wahaibi, Lamya H; Macías, Mario A; Blacque, Olivier; Zondagh, Luke S; Joubert, Jacques; Thamotharan, Subbiah; Percino, María Judith; Mohamed, Ahmed A B; El-Emam, Ali A (2022). Weak Noncovalent Interactions in Three Closely Related Adamantane-Linked 1,2,4-Triazole N-Mannich Bases: Insights from Energy Frameworks, Hirshfeld Surface Analysis, In Silico 11β-HSD1 Molecular Docking and ADMET Prediction. Molecules, 27(21):7403.

Fay, Rachael; Törő, Imre; Schinke, Anna-Lena; Simic, Branko; Schaefer, Jonas V; Dreier, Birgit; Plückthun, Andreas; Holland, Jason P (2022). Sortase-Mediated Site-Specific Conjugation and 89Zr-Radiolabeling of Designed Ankyrin Repeat Proteins for PET. Molecular Pharmaceutics, 19(10):3576-3585.

Spiess, Deborah; Winker, Moritz; Chauveau, Antoine; Abegg, Vanessa Fabienne; Potterat, Olivier; Hamburger, Matthias; Gründemann, Carsten; Simões-Wüst, Ana Paula (2022). Medicinal Plants for the Treatment of Mental Diseases in Pregnancy: An In Vitro Safety Assessment. Planta medica, 88(12):1036-1046.

Martínez-Pizarro, Ainhoa; Leal, Fátima; Holm, Lise Lolle; Doktor, Thomas K; Petersen, Ulrika S S; Bueno, María; Thöny, Beat; Pérez, Belén; Andresen, Brage S; Desviat, Lourdes R (2022). Antisense Oligonucleotide Rescue of Deep-Intronic Variants Activating Pseudoexons in the 6-Pyruvoyl-Tetrahydropterin Synthase Gene. Nucleic Acid Therapeutics, 32(5):378-390.

Nai, Francesco; Nachawati, Raed; Zálešák, František; Wang, Xiang; Li, Yaozong; Caflisch, Amedeo (2022). Fragment Ligands of the m$^{6}$A-RNA Reader YTHDF2. ACS Medicinal Chemistry Letters, 13(9):1500-1509.

Dalle Vedove, Andrea; Cazzanelli, Giulia; Batiste, Laurent; Marchand, Jean-Rémy; Spiliotopoulos, Dimitrios; Corsi, Jessica; D'Agostino, Vito Giuseppe; Caflisch, Amedeo; Lolli, Graziano (2022). Identification of a BAZ2A-Bromodomain Hit Compound by Fragment Growing. ACS Medicinal Chemistry Letters, 13(9):1434-1443.

Spiess, Deborah; Abegg, Vanessa Fabienne; Chauveau, Antoine; Treyer, Andrea; Reinehr, Michael; Oufir, Mouhssin; Duong, Elisa; Potterat, Olivier; Hamburger, Matthias; Simões-Wüst, Ana Paula (2022). Placental Passage of Protopine in an Ex Vivo Human Perfusion System. Planta medica, 87(14):1192-1205.

Sauser, Luca; Kalvoda, Tadeáš; Kavas, Ayça; Rulíšek, Lubomír; Shoshan, Michal S (2022). Cyclic Octapeptides Composed of Two Glutathione Units Outperform the Monomer in Lead Detoxification. ChemMedChem, 17(15):e202200152.

Laitinen, Tuomo; Meili, Theres; Koyioni, Maria; Koutentis, Panayiotis A; Poso, Antti; Hofmann-Lehmann, Regina; Asquith, Christopher R M (2022). Synthesis and evaluation of 1,2,3-dithiazole inhibitors of the nucleocapsid protein of feline immunodeficiency virus (FIV) as a model for HIV infection. Bioorganic & Medicinal Chemistry, 68:116834.

Quirke, Jonathan C K; Sati, Girish C; Sonousi, Amr; Gysin, Marina; Haldimann, Klara; Böttger, Erik C; Vasella, Andrea; Hobbie, Sven N; Crich, David (2022). Structure-Activity Relationships for 5'' Modifications of 4,5-Aminoglycoside Antibiotics. ChemMedChem, 17(13):e202200120.

Scholkmann, Felix; Tsenkova, Roumiana (2022). Changes in Water Properties in Human Tissue after Double Filtration Plasmapheresis-A Case Study. Molecules, 27(12):3947.

Kurz, Christian G; Preuss, Franziska; Tjaden, Amelie; Cusack, Martin; Amrhein, Jennifer Alisa; Chatterjee, Deep; Mathea, Sebastian; Berger, Lena Marie; Berger, Benedict-Tilman; Krämer, Andreas; Weller, Michael; Weiss, Tobias; Müller, Susanne; Knapp, Stefan; Hanke, Thomas (2022). Illuminating the Dark: Highly Selective Inhibition of Serine/Threonine Kinase 17A with Pyrazolo[1,5- a]pyrimidine-Based Macrocycles. Journal of Medicinal Chemistry, 65(11):7799-7817.

Menne, Felix; Schipke, Carola G; Clark, Christopher; Popp, Julius (2022). Long-term stability and age-dependence of six regulatory serum proteins. Biomarkers in Medicine, 16(7):511-521.

Sigel, Astrid; Sigel, Helmut; Sigel, Roland K O (2022). Coordination Chemistry of Nucleotides and Antivirally Active Acyclic Nucleoside Phosphonates, including Mechanistic Considerations. Molecules, 27(9):2625.

Hornemann, Thorsten (2022). Sphingolipids and metabolic disease: Will the real killer please stand up? Molecular Therapy, 30(4):1359-1360.

Göbel, Dominik; Míguez‐Lago, Sandra; Ruedas‐Rama, Maria Jose; Orte, Angel; Campaña, Araceli G; Juricek, Michal (2022). Circularly Polarized Luminescence of [6]Helicenes through Excited-State Intramolecular Proton Transfer. Helvetica Chimica Acta, 105(4):e202100221.

Di Nitto, Cesare; Neri, Dario; Weiss, Tobias; Weller, Michael; De Luca, Roberto (2022). Design and Characterization of Novel Antibody-Cytokine Fusion Proteins Based on Interleukin-21. Antibodies, 11:19.

Tusup, Marina; Kündig, Thomas M; Pascolo, Steve (2022). Epitranscriptomics modifier pentostatin indirectly triggers Toll-like receptor 3 and can enhance immune infiltration in tumors. Molecular Therapy, 30(3):1163-1170.

Müller, Peter; Probst, Benjamin; Spingler, Bernhard; Blacque, Olivier; Alberto, Roger (2022). Polar Substituents Enable Efficient Catalysis for a Class of Cobalt Polypyridyl Hydrogen Evolving Catalysts. Helvetica Chimica Acta, 105(3):e202100237.

Blumberg, Markus; Al-Ameed, Karrar; Eiselt, Erik; Luber, Sandra; Mamat, Constantin (2022). Synthesis of Ionizable Calix[4]arenes for Chelation of Selected Divalent Cations. Molecules, 27(5):1478.

Amiri Rudbari, Hadi; Saadati, Arezoo; Aryaeifar, Mahnaz; Blacque, Olivier; Cuevas-Vicario, Jose V; Cabral, Rui; Raposo, Luis R; Fernandes, Alexandra R (2022). Platinum(II) and Copper(II) complexes of asymmetric halogen-substituted [NNʹO] ligands: Synthesis, characterization, structural investigations and antiproliferative activity. Bioorganic Chemistry, 119:105556.

Naegeli, Hanspeter; Gsell, Corina (2022). "Nano-ghosts": Risk assessment of submicron-sized particles in food biased towards fictional "nano". EXCLI Journal, 21:279-299.

Guillou, Amaury; Nisli, Eda; Klingler, Simon; Linden, Anthony; Holland, Jason P (2022). Photoactivatable Fluorescent Tags for Dual-Modality Positron Emission Tomography Optical Imaging. Journal of Medicinal Chemistry, 65(1):811-823.

Berlowitz, Ilana; O'Shaughnessy, David M; Heinrich, Michael; Wolf, Ursula; Maake, Caroline; Martin-Soelch, Chantal (2022). Teacher plants — Indigenous Peruvian-Amazonian dietary practices as a method for using psychoactives. Journal of Ethnopharmacology, 286:114910.


Shchelik, Inga S; Gademann, Karl (2021). Thiol- and Disulfide-Containing Vancomycin Derivatives Against Bacterial Resistance and Biofilm Formation. ACS Medicinal Chemistry Letters, 12(12):1898-1904.

Mattiat, Johann; Luber, Sandra (2021). Recent Progress in the Simulation of Chiral Systems with Real Time Propagation Methods. Helvetica Chimica Acta, 104(12):e2100154.

Villiger, Lukas; Schmidheini, Lukas; Mathis, Nicolas; Rothgangl, Tanja; Marquart, Kim; Schwank, Gerald (2021). Replacing the SpCas9 HNH domain by deaminases generates compact base editors with an alternative targeting scope. Molecular Therapy : Nucleic Acids, 26:502-510.

Glasauer, Stella M K; Triemer, Therese; Neef, Anne B; Neuhauss, Stephan C F; Luedtke, Nathan W (2021). DNA template strand segregation in developing zebrafish. Cell Chemical Biology, 28(11):1638-1647.e4.

Ni, Ruiqing (2021). Positron Emission Tomography in Animal Models of Alzheimer's Disease Amyloidosis: Translational Implications. Pharmaceuticals, 14(11):1179.

Bassi, Gabriele; Favalli, Nicholas; Pellegrino, Christian; Onda, Yuichi; Scheuermann, Jörg; Cazzamalli, Samuele; Manz, Markus G; Neri, Dario (2021). Specific Inhibitor of Placental Alkaline Phosphatase Isolated from a DNA-Encoded Chemical Library Targets Tumor of the Female Reproductive Tract. Journal of Medicinal Chemistry, 64(21):15799-15809.

Kullak-Ublick, Gerd A (2021). Nukleäre Rezeptoren beim hepatischen und intestinalen Medikamententransport. Drug Research, 71:S13-S14.

Scotti, Francesca; Mou, Linru; Huang, Chen; Booker, Anthony; Weckerle, Caroline; Maake, Caroline; Heinrich, Michael (2021). Treating Chronic Wounds Using Photoactive Metabolites: Data Mining the Chinese Pharmacopoeia for Potential Lead Species. Planta medica, 87(14):1206-1218.

Spiess, Deborah; Abegg, Vanessa Fabienne; Chauveau, Antoine; Treyer, Andrea; Reinehr, Michael; Oufir, Mouhssin; Duong, Elisa; Potterat, Olivier; Hamburger, Matthias; Simões-Wüst, Ana Paula (2021). Retraction: Placental Passage of Humulone and Protopine in an Ex Vivo Human Perfusion System. Planta medica, 87(14):1192-1205.

Moroz-Omori, Elena V; Huang, Danzhi; Kumar Bedi, Rajiv; Cheriyamkunnel, Sherry J; Bochenkova, Elena; Dolbois, Aymeric; Rzeczkowski, Maciej D; Li, Yaozong; Wiedmer, Lars; Caflisch, Amedeo (2021). METTL3 Inhibitors for Epitranscriptomic Modulation of Cellular Processes. ChemMedChem, 16(19):3035-3043.

Rudbari, Hadi Amiri; Saadati, Arezoo; Aryaeifar, Mahnaz; Correia, Isabel; Marques, Fernanda; Blacque, Olivier; Micale, Nicola (2021). Cytotoxic oxidovanadium(IV) complexes of tridentate halogen‐substituted Schiff bases: First dinuclear V(IV) complexes with O → VIV = O → VIV = O core. Bioorganic & Medicinal Chemistry Letters, 49:128285.

Pirrone, Michael G; Hobbie, Sven N; Vasella, Andrea; Böttger, Erik C; Crich, David (2021). Influence of ring size in conformationally restricted ring I analogs of paromomycin on antiribosomal and antibacterial activity. RSC Medicinal Chemistry, 12(9):1585-1591.

Yilmaz, Bahtiyar; Ruckstuhl, Lisa; Müllhaupt, Beat; Magenta, Lorenzo; Kuster, Melanie Harrer; Clerc, Olivier; Torgler, Ralph; Semmo, Nasser (2021). Pilot Sub-Study of the Effect of Hepatitis C Cure by Glecaprevir/Pibrentasvir on the Gut Microbiome of Patients with Chronic Hepatitis C Genotypes 1 to 6 in the Mythen Study. Pharmaceuticals, 14(9):931.

Dolbois, Aymeric; Bedi, Rajiv K; Bochenkova, Elena; Müller, Anna; Moroz-Omori, Elena V; Huang, Danzhi; Caflisch, Amedeo (2021). 1,4,9-Triazaspiro[5.5]undecan-2-one Derivatives as Potent and Selective METTL3 Inhibitors. Journal of Medicinal Chemistry, 64(17):12738-12760.

Dulla, Kalyan; Slijkerman, Ralph; van Diepen, Hester C; Albert, Silvia; Dona, Margo; et al; Zang, Jingjing; Neuhauss, Stephan C F (2021). Antisense oligonucleotide-based treatment of retinitis pigmentosa caused by USH2A exon 13 mutations. Molecular Therapy, 29(8):2441-2455.

Buzzi, Raphael M; Owczarek, Catherine M; Akeret, Kevin; Tester, Andrea; Pereira, Natasha; Butcher, Rebecca; Brügger-Verdon, Valérie; Hardy, Matthew P; Illi, Marlies; Wassmer, Andreas; Vallelian, Florence; Humar, Rok; Hugelshofer, Michael; Buehler, Paul W; Gentinetta, Thomas; Schaer, Dominik J (2021). Modular Platform for the Development of Recombinant Hemoglobin Scavenger Biotherapeutics. Molecular Pharmaceutics, 18(8):3158-3170.

Brenig, Christopher; Mosberger, Leila; Baumann, Katja; Blacque, Olivier; Zelder, Felix (2021). Redox-Neutral Syntheses and Electrochemical Studies of 10-Bromo-Substituted Light-Stable Antivitamin B12 Candidates. Helvetica Chimica Acta, 104:e21000.

Münz, Christian (2021). Natural Killer Cell Responses during Human γ-Herpesvirus Infections. Vaccines, 9(6):655.

Sun, Jiyun; Xiao, Zhiwei; Haider, Ahmed; Gebhard, Catherine; Xu, Hao; Luo, Hai-Bin; Zhang, Han-Ting; Josephson, Lee; Wang, Lu; Liang, Steven H (2021). Advances in Cyclic Nucleotide Phosphodiesterase-Targeted PET Imaging and Drug Discovery. Journal of Medicinal Chemistry, 64(11):7083-7109.

Dharuman, Suresh; Wilt, Laura A; Liu, Jiuyu; Reeve, Stephanie M; Thompson, Carl W; Elmore, John M; Shcherbakov, Dimitri; Lee, Robin B; Böttger, Erik C; Lee, Richard E (2021). Synthesis, antibacterial action, and ribosome inhibition of deoxyspectinomycins. Journal of Antibiotics, 74(6):381-396.

Li, Bei; Chen, Meiling; Aguzzi, Adriano; Zhu, Caihong (2021). The role of macrophage scavenger receptor 1 (Msr1) in prion pathogenesis. Journal of Molecular Medicine, 99(6):877-887.

Le, Ngoc An; Babu, Vipin; Kalt, Martina; Schneider, Lukas; Schumer, Frank; Spingler, Bernhard (2021). Photostable Platinated Bacteriochlorins as Potent Photodynamic Agents. Journal of Medicinal Chemistry, 64(10):6792-6801.

Schabert, Günter; Haase, Robert; Parris, Jaclyn; Pala, Laura; Hery-Barranco, Adrian; Spingler, Bernhard; Spitz, Urs (2021). New Crystalline Salts of Nicotinamide Riboside as Food Additives. Molecules, 26(9):2729.

Cumming, Paul; Scheidegger, Milan; Dornbierer, Dario; Palner, Mikael; Quednow, Boris B; Martin-Soelch, Chantal (2021). Molecular and Functional Imaging Studies of Psychedelic Drug Action in Animals and Humans. Molecules, 26(9):2451.

Liberini, Virginia; Laudicella, Riccardo; Capozza, Martina; Huellner, Martin W; Burger, Irene A; Baldari, Sergio; Terreno, Enzo; Deandreis, Désirée (2021). The Future of Cancer Diagnosis, Treatment and Surveillance: A Systemic Review on Immunotherapy and Immuno-PET Radiotracers. Molecules, 26(8):2201.

Jäger, Levy; Senn, Oliver; Rosemann, Thomas; Plate, Andreas (2021). Awareness, Attitudes and Clinical Practices Regarding Human Papillomavirus Vaccination among General Practitioners and Pediatricians in Switzerland. Vaccines, 9(4):332.

Waltenspühl, Yann; Ehrenmann, Janosch; Klenk, Christoph; Plückthun, Andreas (2021). Engineering of Challenging G Protein-Coupled Receptors for Structure Determination and Biophysical Studies. Molecules, 26(5):1465.

Hassell‐Hart, Storm; Picaud, Sarah; Lengacher, Raphael; Csucker, Joshua; Millet, Regis; Gasser, Gilles; Alberto, Roger; Maple, Hannah; Felix, Robert; Leśnikowski, Zbigniew J; Stewart, Helen J S; Chevassut, Timothy J; Morley, Simon; Filippakopoulos, Panagis; Spencer, John (2021). Probing BRD Inhibition Substituent Effects in Bulky Analogues of (+)‐JQ1. Helvetica Chimica Acta, 104(3):e2000214.

Padrutt, Roxane; Babu, Vipin; Klingler, Simon; Kalt, Martina; Schumer, Frank; Anania, Maria I; Schneider, Lukas; Spingler, Bernhard (2021). Highly Phototoxic Transplatin‐Modified Distyryl‐BODIPY Photosensitizers for Photodynamic Therapy. ChemMedChem, 16(4):694-701.

Earley, Daniel F; Guillou, Amaury; van der Born, Dion; Poot, Alex J; Holland, Jason P (2021). Microfluidic Preparation of 89Zr-Radiolabelled Proteins by Flow Photochemistry. Molecules, 26(3):764.

Wirsching, Hans-Georg; Roth, Patrick; Weller, Michael (2021). A vasculature-centric approach to developing novel treatment options for glioblastoma. Expert Opinion on Therapeutic Targets, 25(2):87-100.

Sonousi, Amr; Quirke, Jonathan C K; Waduge, Prabuddha; Janusic, Tanja; Gysin, Marina; Haldimann, Klara; Xu, Shan; Hobbie, Sven N; Sha, Su-Hua; Schacht, Jochen; Chow, Christine S; Vasella, Andrea; Böttger, Erik C; Crich, David (2021). An Advanced Apralog with Increased in vitro and in vivo Activity toward Gram-negative Pathogens and Reduced ex vivo Cochleotoxicity. ChemMedChem, 16(2):335-339.

Hou, Lu; Rong, Jian; Haider, Ahmed; Ogasawara, Daisuke; Varlow, Cassis; Schafroth, Michael A; Mu, Linjing; Gan, Jiefeng; Xu, Hao; Fowler, Christopher J; Zhang, Ming-Rong; Vasdev, Neil; Ametamey, Simon; Cravatt, Benjamin F; Wang, Lu; Liang, Steven H (2021). Positron Emission Tomography Imaging of the Endocannabinoid System: Opportunities and Challenges in Radiotracer Development. Journal of Medicinal Chemistry, 64(1):123-149.

Zabulica, Mihaela; Srinivasan, Raghuraman C; Akcakaya, Pinar; Allegri, Gabriella; Bestas, Burcu; Firth, Mike; Hammarstedt, Christina; Jakobsson, Tomas; Jakobsson, Towe; Ellis, Ewa; Jorns, Carl; Makris, Georgios; Scherer, Tanja; Rimann, Nicole; van Zuydam, Natalie R; Gramignoli, Roberto; Forslöw, Anna; Engberg, Susanna; Maresca, Marcello; Rooyackers, Olav; Thöny, Beat; Häberle, Johannes; Rosen, Barry; Strom, Stephen C (2021). Correction of a urea cycle defect after ex vivo gene editing of human hepatocytes. Molecular Therapy, 29(5):1903-1917.


He, Yingfang; Whitehead, David M; Briard, Emmanuelle; Numao, Shin; Mu, Linjing; Schibli, Roger; Ametamey, Simon M; Auberson, Yves P (2020). Evaluation of 5H-Thiazolo[3,2-α]pyrimidin-5-ones as Potential GluN2A PET Tracers. ChemMedChem, 15(24):2448-2461.

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Arnhold, Franziska S; Linden, Anthony; Heimgartner, Heinz (2015). Synthesis of Aib- and Phe(2Me)-Containing Cyclopentapeptides. Helvetica Chimica Acta, 98(2):155-178.

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Stadlbauer, Ulrike; Meyer, Urs (2015). Developmental Neuroimmune Mechanisms in Schizophrenia. In: Lipina, Tatiana; Roder, John. Drug Discovery for Schizophrenia. Cambridge: Royal Society of Chemistry, 46-69.

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Chen, Yi; Lehto, Erja; Uebelhart, Peter; Linden, Anthony; Hansen, Hans-Jürgen (2015). Excursion to the World of Heptacyclic Compounds Made of Azulenes and Acetylenedicarboxylates. Helvetica Chimica Acta, 98(7):913-937.

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Chiotellis, Aristeidis; Muller, Adrienne; Mu, Linjing; Keller, Claudia; Schibli, Roger; Krämer, Stefanie D; Ametamey, Simon M (2014). Synthesis and biological evaluation of (18)F-labeled Fluoroethoxy tryptophan analogues as potential PET tumor imaging agents. Molecular Pharmaceutics, 11(11):3839-3851.

Schwendener, Reto A (2014). Liposomes as vaccine delivery systems: A review of the recent advances. Therapeutic Advances in Vaccines, 2(6):159-182.

Mandhapati, Appi Reddy; Shcherbakov, Dimitri; Duscha, Stefan; Vasella, Andrea; Böttger, Erik C; Crich, David (2014). Importance of the 6'-hydroxy group and its configuration for apramycin activity. ChemMedChem, 9(9):2074-2083.

Cavkaytar, Ozlem; Akdis, Cezmi A; Akdis, Mübeccel (2014). Modulation of immune responses by immunotherapy in allergic diseases. Current Opinion in Pharmacology, 17:30-37.

Leonidova, Anna; Pierroz, Vanessa; Adams, Luke A; Barlow, Nicholas; Ferrari, Stefano; Graham, Bim; Gasser, Gilles (2014). Enhanced Cytotoxicity through Conjugation of a "Clickable" Luminescent Re(I) Complex to a Cell-Penetrating Lipopeptide. ACS Medicinal Chemistry Letters, 5(7):809-814.

Joshi, Tanmaya; Pierroz, Vanessa; Ferrari, Stefano; Gasser, Gilles (2014). Bis(dipyridophenazine)(2-(2'-pyridyl)pyrimidine-4-carboxylic acid)ruthenium(II) hexafluorophosphate: a lesson in stubbornness. ChemMedChem, 9(7):1419-1427.

Gebert, Andreas; Jasiński, Marcin; Mlostoń, Grzegorz; Heimgartner, Heinz (2014). Reduction of Thiocarbonyl Compounds with Lithium Diisopropylamide. Helvetica Chimica Acta, 97(7):931-938.

Asquith, Christopher R M; Meli, Marina L; Konstantinova, Lidia S; Laitinen, Tuomo; Peräkylä, Mikael; Poso, Antti; Rakitin, Oleg A; Allenspach, Karin; Hofmann-Lehmann, Regina; Hilton, Stephen T (2014). Evaluation of the antiviral efficacy of bis[1,2]dithiolo[1,4]thiazines and bis[1,2]dithiolopyrrole derivatives against the nucelocapsid protein of the Feline Immunodeficiency Virus (FIV) as a model for HIV infection. Bioorganic & Medicinal Chemistry Letters, 24(12):2640-2644.

Botter, Sander M; Neri, Dario; Fuchs, Bruno (2014). Recent advances in osteosarcoma. Current Opinion in Pharmacology, 16:15-23.

Gianferrara, Teresa; Spagnul, Cinzia; Alberto, Roger; Gasser, Gilles; Ferrari, Stefano; Pierroz, Vanessa; Bergamo, Alberta; Alessio, Enzo (2014). Towards matched pairs of porphyrin-Re(I) /(99m) Tc(I) conjugates that combine photodynamic activity with fluorescence and radio imaging. ChemMedChem, 9(6):1231-1237.

Seeger, Stefan (2014). Future pharmaceutical research: The need to look beyond science. Future Medicinal Chemistry, 6(7):721-723.

Khlebnikov, Alexander F; Konev, Alexander S; Virtsev, Alexander A; Yufit, Dmitri S; Mlostoń, Grzegorz; Heimgartner, Heinz (2014). Concerted vs. Non-Concerted 1,3-Dipolar Cycloadditions of Azomethine Ylides to Electron-Deficient Dialkyl 2,3-Dicyanobut-2-enedioates. Helvetica Chimica Acta, 97:453-470.

Balabanov, S; Braig, M; Brümmendorf, T H (2014). Current aspects in resistance against tyrosine kinase inhibitors in chronic myelogenous leukemia. Drug Discovery Today: Technologies, 11:89-99.

Forster, Simon P; Stegmaier, Julia; Spycher, Rene; Seeger, Stefan (2014). Virtual pharmaceutical companies: Collaborating flexibly in pharmaceutical development. Drug Discovery Today, 19(3):348-355.

Brokamp, Renate; Bergmann, Bärbel; Müller, Ingrid B; Bienz, Stefan (2014). Stereoselective preparation of pyridoxal 1,2,3,4-tetrahydro-β-carboline derivatives and the influence of their absolute and relative configuration on the proliferation of the malaria parasite Plasmodium falciparum. Bioorganic & Medicinal Chemistry, 22(6):1832-1837.

Gallego-Villar, Lorena; Viecelli, Hiu Man; Pérez, Belén; Harding, Cary O; Ugarte, Magdalena; Thöny, Beat; Desviat, Lourdes R (2014). A sensitive assay system to test antisense oligonucleotides for splice suppression therapy in the mouse liver. Molecular Therapy : Nucleic Acids, 3:e193.

von Rechenberg, Brigitte (2014). Animal models in bone repair. Drug Discovery Today: Disease Models, 13:23-27.

Rubbiani, Riccardo; Zehnder, Thomas N; Mari, Cristina; Blacque, Olivier; Venkatesan, Koushik; Gasser, Gilles (2014). Anticancer Profile of a Series of Gold(III) (2-phenyl)pyridine Complexes. ChemMedChem, 9(12):2781-2790.

Zupo, Valerio; Jüttner, Friedrich; Maibam, Chingoileima; Butera, Emanuela; Blom, Judith (2014). Apoptogenic Metabolites in Fractions of the Benthic Diatom Cocconeis scutellum parva. Marine Drugs, 12(1):547-567.

Portmann, Cyril; Sieber, Simon; Wirthensohn, Silvan; Blom, Judith F; Da Silva, Laeticia; Baudat, Emilie; Kaiser, Marcel; Brun, Reto; Gademann, Karl (2014). Balgacyclamides, Antiplasmodial Heterocyclic Peptides fromMicrocystis aeruguinosaEAWAG 251. Journal of natural products, 77(3):557-562.

Vavricka, Stephan R; Scharl, Michael; Gubler, Martin; Rogler, Gerhard (2014). Biologics for extraintestinal manifestations of IBD. Current Drug Targets, 15(11):1064-73.

Tonder, M; Weller, M; Eisele, G; Roth, P (2014). Carboplatin and Etoposide in Heavily Pretreated Patients with Progressive High-Grade Glioma. Chemotherapy, 60(5-6):375-378.

Pauli, Denise; Bienz, Stefan (2014). Development of a new linker for the solid-phase synthesis of N-hydroxylated and N-methylated secondary amines. Tetrahedron, 70(6):1348-1356.

Zhao, Hongtao; Gartenmann, Lisa; Dong, Jing; Spiliotopoulos, Dimitrios; Caflisch, Amedeo (2014). Discovery of BRD4 bromodomain inhibitors by fragment-based high-throughput docking. Bioorganic & Medicinal Chemistry Letters, 24(11):2493-2496.

Zhao, Hongtao; Caflisch, Amedeo (2014). Discovery of dual ZAP70 and Syk kinases inhibitors by docking into a rare C-helix-out conformation of Syk. Bioorganic & Medicinal Chemistry Letters, 24(6):1523-1527.

Mori, Mattia; Moraca, Francesca; Deodato, Davide; Ferraris, Davide M; Selchow, Petra; Sander, Peter; Rizzi, Menico; Botta, Maurizio (2014). Discovery of the first potent and selective Mycobacterium tuberculosis Zmp1 inhibitor. Bioorganic & Medicinal Chemistry Letters, 24(11):2508-2511.

Kaufmann, Kerstin B; Chiriaco, Maria; Siler, Ulrich; Finocchi, Andrea; Reichenbach, Janine; Stein, Stefan; Grez, Manuel (2014). Gene therapy for chronic granulomatous disease: current status and future perspectives. Current Gene Therapy, 14(6):447-60.

Spiliotopoulos, Dimitrios; Caflisch, Amedeo (2014). Molecular Dynamics Simulations of Bromodomains Reveal Binding-Site Flexibility and Multiple Binding Modes of the Natural Ligand Acetyl-Lysine. Israel Journal of Chemistry, 54(8-9):1084-1092.

Kränkel, Nicolle; Lüscher, Thomas F; Landmesser, Ulf (2014). Novel insights into vascular repair mechanisms. Current Pharmaceutical Design, 20(14):2430-2438.

Myburgh, Renier; Cherpin, Ophélie; Schlaepfer, Erika; Rehrauer, Hubert; Speck, Roberto F; Krause, Karl-Heinz; Salmon, Patrick (2014). Optimization of critical hairpin features allows miRNA-based gene knockdown upon single-copy transduction. Molecular Therapy : Nucleic Acids, 3:e207.

Unzue, Andrea; Dong, Jing; Lafleur, Karine; Zhao, Hongtao; Frugier, Emilie; Caflisch, Amedeo; Nevado, Cristina (2014). Pyrrolo[3,2-b]quinoxaline derivatives as types I1/2 and II Eph tyrosine kinase inhibitors: structure-based design, synthesis, and in vivo validation. Journal of Medicinal Chemistry, 57(15):6834-6844.

Engler, Anna; Niederer, Fabienne; Klein, Kerstin; Gay, Renate E; Kyburz, Diego; Camici, Giovanni G; Gay, Steffen; Ospelt, Caroline (2014). SIRT6 regulates the cigarette smoke-induced signalling in rheumatoid arthritis synovial fibroblasts. Journal of Molecular Medicine, 92(7):757-767.

Shalaby, Tarek; Fiaschetti, Giulio; Baumgartner, Martin; Grotzer, Michael A (2014). Significance and therapeutic value of miRNAs in embryonal neural tumors. Molecules, 19(5):5821-5862.

Lambrigger-Steiner, C; Simões-Wüst, Ana Paula; Kuck, A; Fürer, K; Hamburger, M; von Mandach, U (2014). Sleep quality in pregnancy during treatment with Bryophyllum pinnatum: An observational study. Phytomedicine, 21(5):753-757.

Arnhold, Franziska S; Linden, Anthony; Heimgartner, Heinz (2014). Synthesis of Z-Protected Aib- and Phe(2Me)-Containing Pentapeptides and Their Crystal Structures. Helvetica Chimica Acta, 97(5):619-645.

Frei, Angelo; Rubbiani, Riccardo; Tubafard, Solmaz; Blacque, Olivier; Anstätt, Philipp; Felgenträger, Ariane; Maisch, Tim; Spiccia, Leone; Gasser, Gilles (2014). Synthesis, Characterization and Biological Evaluation of New Ru(II) Polypyridyl Photosensitizers for Photodynamic Therapy. Journal of Medicinal Chemistry, 57(17):7280-7292.

Chen, Weiwei; Matsushita, Takahiko; Shcherbakov, Dimitri; Boukari, Heithem; Vasella, Andrea; Böttger, Erik C; Crich, David (2014). Synthesis, antiribosomal and antibacterial activity of 4'-O-glycopyranosyl paromomycin aminoglycoside antibiotics. MedChemComm, 5:1179-1187.

Dal Cero, Maja; Saller, Reinhard; Weckerle, Caroline S (2014). The use of the local flora in Switzerland: A comparison of past and recent medicinal plant knowledge. Journal of Ethnopharmacology, 151(1):253-264.


Shalaby, Tarek; Fiaschetti, Giulio; Nagasawa, Kazuo; Shin-Ya, Kazuo; Baumgartner, Martin; Grotzer, Michael (2013). G-quadruplexes as potential therapeutic targets for embryonal tumors. Molecules, 18(10):12500-12537.

Mitchell, Ruth; Trück, Johannes; Pollard, Andrew J (2013). Use of the 13-valent pneumococcal conjugate vaccine in children and adolescents aged 6 - 17 years. Expert Opinion on Biological Therapy, 13(10):1451-1465.

Stoykova, Svetlana A; Linden, Anthony; Heimgartner, Heinz (2013). Highly Constrained Linear Oligopeptides Containing Heterocyclic alpha-Amino Carboxylic Acids. Helvetica Chimica Acta, 96(9):1714-1732.

Shi, Jungxing; Linden, Anthony; Heimgartner, Heinz (2013). Reactions of acid Chlorides/Ketenes with 2-substituted 4,5-Dihydro-4,4-dimethyl-1,3-thiazoles: Formation of Penam derivatives. Helvetica Chimica Acta, 96(8):1462-1481.

Schmidt, Jasmin; Patora-Komisarska, Kristina; Moehle, Kerstin; Obrecht, Daniel; Robinson, John A (2013). Structural studies of β-hairpin peptidomimetic antibiotics that target LptD in Pseudomonas sp. Bioorganic & Medicinal Chemistry, 21(18):5806-5810.

Ali, Korany A; Ragab, Eman A; Mlostoń, Grzegorz; Celeda, Malgorzata; Linden, Anthony; Heimgartner, Heinz (2013). Unexpected reaction course of 3-Amino-5-aryl-1H-pyrazoles with Dialkyl Dicyanofumarates. Helvetica Chimica Acta, 96(4):633-643.

Pieczonka, Adam M; Ciepielowski, Krzysztof; Cebulska, Zofia; Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (2013). New selenosemicarbazides derived from imidazole-based carbohydrazides. Helvetica Chimica Acta, 96(3):397-407.

Robinson, John A (2013). Max Bergmann lecture protein epitope mimetics in the age of structural vaccinology. Journal of Peptide Science, 19(3):127-140.

Lacher, Markus D; Provenzano, Maurizio (2013). Cancer T cell immunotherapy with bispecific antibodies and chimeric antigen receptors. Recent Patents on Anti-Cancer Drug Discovery, 8(3):239-254.

Uchiyama, Satoshi; Andreoni, Federica; Zürcher, Claudia; Schilcher, Katrin; Ender, Miriam; Madon, Jerzy; Matt, Ulrich; Ghosh, Partho; Nizet, Victor; Schuepbach, Reto A; Zinkernagel, Annelies S (2013). Coiled-coil irregularities of the M1 protein structure promote M1-fibrinogen interaction and influence group A Streptococcus host cell interactions and virulence. Journal of Molecular Medicine, 91(7):861-869.

Benz, Sebastian; Noetzli, Sarah; Siegel, Jay; Eberli, Daniel; Jessen, Henning Jacob (2013). Controlled oxygen release from pyridone endoperoxides promotes cell survival under anoxic conditions. Journal of Medicinal Chemistry, 56(24):10171-10182.

Friedrich, Katrin; Hanauer, Jan R H; Prüfer, Steffen; Münch, Robert C; Völker, Iris; Filippis, Christodoulos; Jost, Christian; Hanschmann, Kay-Martin; Cattaneo, Roberto; Peng, Kah-Whye; Plückthun, Andreas; Buchholz, Christian J; Cichutek, Klaus; Mühlebach, Michael D (2013). DARPin-targeting of measles virus: unique bispecificity, effective oncolysis, and enhanced safety. Molecular Therapy, 21(4):849-859.

Zhao, Hongtao; Caflisch, Amedeo (2013). Discovery of ZAP70 inhibitors by high-throughput docking into a conformation of its kinase domain generated by molecular dynamics. Bioorganic & Medicinal Chemistry Letters, 23(20):5721-5726.

Klein, Kerstin; Gay, Steffen (2013). Epigenetic modifications in rheumatoid arthritis, a review. Current Opinion in Pharmacology, 13(3):420-425.

Landmesser, Thomas; Linden, Anthony; Hansen, Hans-Jürgen (2013). From blue Azulenes to blue Heptalenes - new strongly polarized π-convertible heptalenes. Helvetica Chimica Acta, 96(10):1851-1893.

Patra, Malay; Ingram, Katrin; Leonidova, Anna; Pierroz, Vanessa; Ferrari, Stefano; Robertson, Murray N; Todd, Matthew H; Keiser, Jennifer; Gasser, Gilles (2013). In vitro metabolic profile and in vivo antischistosomal activity studies of (η(6)-Praziquantel)Cr(CO)3 derivatives. Journal of Medicinal Chemistry, 56(22):9192-9198.

Kummer, Lutz; Hsu, Chia-Wen; Dagliyan, Onur; Macnevin, Christopher; Kaufholz, Melanie; Zimmermann, Bastian; Dokholyan, Nikolay V; Hahn, Klaus M; Plückthun, Andreas (2013). Knowledge-based design of a biosensor to quantify localized ERK activation in living cells. Chemistry & Biology, 20(6):847-856.

Zobi, Fabio; Quaroni, Luca; Santoro, Giuseppe; Zlateva, Theodora; Blacque, Olivier; Sarafimov, Blagoj; Schaub, Marcus C; Bogdanova, Anna Yu (2013). Live-fibroblast IR imaging of a cytoprotective PhotoCORM Activated with Visible Light. Journal of Medicinal Chemistry, 56(17):6719-6731.

Tomašković, Linda; Komac, Marijana; Makaruha Stegić, Oresta; Munić, Vesna; Ralić, Jovica; Stanić, Barbara; Banjanac, Mihailo; Marković, Stribor; Hrvačić, Boška; Čipčić Paljetak, Hana; Padovan, Jasna; Glojnarić, Ines; Eraković Haber, Vesna; Mesić, Milan; Merćep, Mladen (2013). Macrolactonolides: a novel class of anti-inflammatory compounds. Bioorganic & Medicinal Chemistry, 21(1):321-332.

Monigatti, Martina; Bussmann, Rainer W; Weckerle, Caroline S (2013). Medicinal plant use in two Andean communities located at different altitudes in the Bolívar Province, Peru. Journal of Ethnopharmacology, 145(2):450-464.

Jarzabek, Monika A; Sweeney, Kieron J; Evans, Rhys L; Jacobs, Andreas H; Stupp, Roger; O'Brien, Donncha; Berger, Mitchel S; Prehn, Jochen H M; Byrne, Annette T (2013). Molecular imaging in the development of a novel treatment paradigm for glioblastoma (GBM): an integrated multidisciplinary commentary. Drug Discovery Today, 18(21-22):1052-1066.

Jacomella, Vincenzo; Corti, Natascia; Husmann, Marc (2013). Novel anticoagulants in the therapy of peripheral arterial and coronary artery disease. Current Opinion in Pharmacology, 13(2):294-300.

Gerber, Philipp A; Gouni-Berthold, Ioanna; Berneis, Kaspar (2013). Omega-3 fatty acids: role in metabolism and cardiovascular disease. Current Pharmaceutical Design, 19(17):3074-3093.

Lafleur, Karine; Dong, Jing; Huang, Danzhi; Caflisch, Amedeo; Nevado, Cristina (2013). Optimization of inhibitors of the tyrosine kinase EphB4. 2. Cellular potency improvement and binding mode validation by X-ray crystallography. Journal of Medicinal Chemistry, 56(1):84-96.

Viel, Thomas; Monfared, Parisa; Schelhaas, Sonja; Fricke, Inga B; Kuhlmann, Michael T; Fraefel, Cornel; Jacobs, Andreas H (2013). Optimizing Glioblastoma Temozolomide chemotherapy employing Lentiviral-based anti-MGMT shRNA technology. Molecular Therapy, 21(3):570-579.

Corti, Natascia; Rudiger, Alain; Chiesa, Alessandro; Marti, Isabelle; Jetter, Alexander; Rentsch, Katharina; Müller, Daniel; Béchir, Markus; Maggiorini, Marco (2013). Pharmacokinetics of daily daptomycin in critically ill patients undergoing continuous renal replacement therapy. Chemotherapy, 59(2):143-151.

Betschart, Cornelia; von Mandach, Ursula; Seifert, Burkhardt; Scheiner, David; Perucchini, Daniele; Fink, Daniel; Geissbühler, Verena (2013). Randomized, double-blind placebo-controlled trial with Bryophyllum pinnatum versus placebo for the treatment of overactive bladder in postmenopausal women. Phytomedicine, 20(3-4):351-358.

Scharl, Michael; Vavricka, Stephan R; Rogler, Gerhard (2013). Review: new anti-cytokines for IBD: what is in the pipeline? Current Drug Targets, 14(12):1405-1420.

Tarasava, K; Johannsen, S; Freisinger, Eva (2013). Solution structure of the circular γ-domain analog from the wheat metallothionein Ec-1. Molecules, 18:14414-14429.

Huang, Danzhi; Rossini, Emanuele; Steiner, Sandra; Caflisch, Amedeo (2013). Structured water molecules in the binding site of bromodomains can be displaced by cosolvent. ChemMedChem, 9(3):573-579.

Chiotellis, Aristeidis; Mu, Linjing; Müller, Adrienne; Selivanova, Svetlana V; Keller, Claudia; Schibli, Roger; Krämer, Stefanie D; Ametamey, Simon M (2013). Synthesis and biological evaluation of (18)F-labeled fluoropropyl tryptophan analogs as potential PET probes for tumor imaging. European journal of medicinal chemistry, 70C:768-780.

Maillefer-El Houar, Sarah; Uebelhart, Peter; Linden, Anthony; Hansen, Hans-Jürgen (2013). Synthesis and characterization of new Heptalenes with extended π-systems attached to them. Helvetica Chimica Acta, 96(8):1488-1541.

Moll, Solange; Chaykovska, Lyubov; Meier, Matthias; Budd, David C; Formentini, Ivan; Pomposiello, Silvia; Prunotto, Marco (2013). Targeting the epithelial cells in fibrosis: a new concept for an old disease. Drug Discovery Today, 18(11-12):582-591.

Schmid, Corina A; Craig, Vanessa J; Müller, Anne; Flori, Michael (2013). The role of microRNAs in the pathogenesis and treatment of hematopoietic malignancies. Current Pharmaceutical Design, 19(7):1201-1210.

Harrow, Ian; Filsell, Wendy; Woollard, Peter; Dix, Ian; Braxtenthaler, Michael; Gedye, Richard; Hoole, David; Kidd, Richard; Wilson, Jabe; Rebholz-Schuhmann, Dietrich (2013). Towards virtual know ledge broker services for semantic integration of life science literature and data sources. Drug Discovery Today, 18(9-10):428-434.

Antic, Milos; Distler, Jörg H W; Distler, Oliver (2013). Treating skin and lung fibrosis in systemic sclerosis: a future filled with promise? Current Opinion in Pharmacology, 13(3):455-462.

Schmid, Fabian; Jessen, Henning Jacob; Burch, Patrick; Gademann, Karl (2013). Truncated militarinone fragments identified by total chemical synthesis induce neurite outgrowth. MedChemComm, 4(1):135-139.

Fürer, Karin; Raith, Melanie; Brenneisen, Rudolf; Mennet, Monica; Simões-Wüst, Ana Paula; von Mandach, Ursula; Hamburger, Matthias; Potterat, Olivier (2013). Two new flavonol glycosides and a metabolite profile of bryophyllum pinnatum, a phytotherapeutic used in obstetrics and gynaecology. Planta medica, 79(16):1565-1571.

Uehleke, B; Müller, J; Stange, R; Kelber, O; Melzer, J (2013). Willow bark extract STW 33-I in the long-term treatment of outpatients with rheumatic pain mainly osteoarthritis or back pain. Phytomedicine, 20(11):980-984.


Stoykova, Svetlana A; Linden, Anthony; Heimgartner, Heinz (2012). Synthesis of Aib-Pro Oligopeptides by repeated Azirine coupling with the Aib-Pro synthon. Helvetica Chimica Acta, 95(8):1325-1350.

Gebert, Andreas; Barth, Max; Linden, Anthony; Widmer, Ulrich; Heimgartner, Heinz (2012). Novel Synthesis of 2-Alkylquinolizinium-1-olates and their 1,3-Dipolar Cycloaddition reactions with Acetylenes. Helvetica Chimica Acta, 95(5):737-760.

Buadze, Anna; Kaiser, S; Stohler, R; Roessler, W; Seifritz, E; Fusar-Poli, P; Liebrenz, M (2012). Patient's perceptions of the cannabis-psychosis link--a systematic review. Current Pharmaceutical Design, 18:5105-5112.

Mlostoń, G; Urbaniak, K; Wojciechowska, A; Linden, Anthony; Heimgartner, H (2012). Unexpected course of the reaction of 2-Unsubstituted 1H-Imidazole 3-Oxides with Ethyl Acrylate. Helvetica Chimica Acta, 95(4):577-585.

Schwarzenbach, Michael; Erismann, Peter; Blättler, Gerhard; Barmettler, Trix (2012). Sapperlot! Mundarten der Schweiz 8.3 - 25.8.2012 : Eine Ausstellung der Schweizerischen Nationalbibliothek und des Phonogrammarchivs der Universität Zürich. Bern: Nationalbibliothek.

Eigeldinger-Berthou, Sylvie; Buntschu, Patrick; Flück, Martin; Frobert, Aurélien; Ferrié, Céline; Carrel, Thierry P; Tevaearai, Hendrik T; Kadner, Alexander (2012). Electric pulses augment reporter gene expression in the beating heart. Journal of Gene Medicine, 14(3):191-203.

Curt, Armin (2012). Human neural stem cells in chronic spinal cord injury. Expert Opinion on Biological Therapy, 12(3):271-273.

Pieczonka, A M; Mlostoń, G; Heimgartner, H (2012). Synthesis of Bis-Heterocyclic 1H-Imidazole 3-Oxides from 3-Oxido-1H-imidazole-4-carbohydrazides. Helvetica Chimica Acta, 95(3):404-414.

Obrecht, Daniel; Chevalier, Eric; Moehle, Kerstin; Robinson, John A (2012). β-Hairpin protein epitope mimetic technology in drug discovery. Drug Discovery Today: Technologies, 9(1):e63-e69.

Abou-Hadeed, Khaled; Molnar, Zoltàn A; Göksaltık, Pinar; Kunz, Roland W; Linden, Anthony; Hansen, Hans-Jürgen (2012). A new alkylation method for heptalene-4,5-dicarboxylates and of one of their pseudoester forms. Helvetica Chimica Acta, 95(6):885-921.

Weckerle, Caroline S; Cabras, Stefano; Castellanos, Maria Eugenia; Leonti, Marco (2012). An imprecise probability approach for the detection of over and underused taxonomic groups with the Campania (Italy) and the Sierra Popoluca (Mexico) medicinal flora. Journal of Ethnopharmacology, 142(1):259-264.

Schuler, V; Suter, K; Fürer, K; Eberli, D; Horst, M; Betschart, C; Brenneisen, R; Hamburger, M; Mennet, M; Schnelle, M; Simões-Wüst, Ana Paula; von Mandach, U (2012). Bryophyllum pinnatum inhibits detrusor contractility in porcine bladder strips - a pharmacological study towards a new treatment option of overactive bladder. Phytomedicine, 19(10):947-951.

Millan, Mark J; Agid, Yves; Brüne, Martin; Bullmore, Edward T; Carter, Cameron S; Clayton, Nicola S; Connor, Richard; Davis, Sabrina; Deakin, Bill; DeRubeis, Robert J; Dubois, Bruno; Geyer, Mark A; Goodwin, Guy M; Gorwood, Philip; Jay, Thérèse M; Joëls, Marian; Mansuy, Isabelle M; Meyer-Lindenberg, Andreas; Murphy, Declan; Rolls, Edmund; Saletu, Bernd; Spedding, Michael; Sweeney, John; Whittington, Miles; Young, Larry J (2012). Cognitive dysfunction in psychiatric disorders: characteristics, causes and the quest for improved therapy. Nature Reviews. Drug Discovery, 11(2):141-168.

Visser, Pieter Jelle; Wolf, Henrike; Frisoni, Giovanni; Gertz, Hermann-Josef (2012). Disclosure of Alzheimer's disease biomarker status in subjects with mild cognitive impairment. Biomarkers in Medicine, 6(4):365-368.

Patra, Malay; Ingram, Katrin; Pierroz, Vanessa; Ferrari, Stefano; Spingler, Bernhard; Keiser, Jennifer; Gasser, Gilles (2012). Ferrocenyl Derivatives of the Anthelmintic Praziquantel: Design, Synthesis, and Biological Evaluation. Journal of Medicinal Chemistry, 55(20):8790-8798.

Laimbacher, Andrea S; Esteban, Laura E; Castello, Alejandro A; Abdusetir Cerfoglio, Juan C; Argüelles, Marcelo H; Glikmann, Graciela; D'Antuono, Alejandra; Mattion, Nora; Berois, Mabel; Arbiza, Juan; Hilbe, Monika; Schraner, Elisabeth M; Seyffert, Michael; Dresch, Christiane; Epstein, Alberto L; Ackermann, Mathias; Fraefel, Cornel (2012). HSV-1 amplicon vectors launch the production of heterologous Rotavirus-like particles and induce Rotavirus-specific immune responses in mice. Molecular Therapy, 20(9):1810-1820.

Rebeaud, Fabien; Bachmann, Martin F (2012). Immunization strategies for Clostridium difficile infections. Expert Review of Vaccines, 11(4):469-479.

Pedersen, S J; Bhatia, V K; Jurt, S; Paulsson, J F; Pedersen, M H; Jorgensen, R; Holst, B; Stamou, D; Vrang, N; Zerbe, O; Jensen, K J (2012). Improving membrane binding as a design strategy for amphipathic peptide hormones: 2-helix variants of PYY3-36. Journal of Peptide Science, 18(9):579-587.

Klingenberg, Roland; Lüscher, Thomas F (2012). Inflammation in coronary artery disease and acute myocardial infarction - is the stage set for novel therapies? Current Pharmaceutical Design, 18(28):4358-4369.

Daud, A; Soon, C; Dummer, R; Eggermont, A M M; Hwu, W J; Grob, J J; Garbe, C; Hauschild, A (2012). Management of pegylated interferon alpha toxicity in adjuvant therapy of melanoma. Expert Opinion on Biological Therapy, 12(8):1087-1099.

Pieczonka, Adam M; Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (2012). New Optically Active Bis-Heterocycles Derived from (S)-Proline. Helvetica Chimica Acta, 95(9):1521-1530.

Benden, Christian; Danziger-Isakov, Lara; Faro, Albert (2012). New developments in treatment after lung transplantation. Current Pharmaceutical Design, 18(5):737-746.

Uehleke, B; Schaper, S; Dienel, A; Schlaefke, S; Stange, R (2012). Phase II trial on the effects of Silexan in patients with neurasthenia, post-traumatic stress disorder or somatization disorder. Phytomedicine, 19(8-9):665-671.

Leonti, Marco; Cabras, Stefano; Castellanos, Maria Eugenia; Weckerle, Caroline S (2012). Reply to the commentary: “Regression residual vs. Bayesian analysis of medicinal floras”. Journal of Ethnopharmacology, 139(3):695-697.

Şafak, Cihat; Gündüz, Miyase Gözde; İlhan, Sevil Özger; Şimşek, Rahime; İşli, Fatma; Yıldırım, Şeniz; Fincan, Gökçe Sevim Öztürk; Sarıoğlu, Yusuf; Linden, Anthony (2012). Synthesis and Myorelaxant activity of fused 1,4-Dihydropyridines on isolated rabbit gastric fundus. Drug Development Research, 73(6):332-342.

Milicevic Sephton, Selena; Mu, Linjing; Schweizer, W Bernd; Schibli, Roger; Krämer, Stefanie D; Ametamey, Simon M (2012). Synthesis and evaluation of novel α-fluorinated (E)-3-((6-methylpyridin-2-yl)ethynyl)cyclohex-2-enone-O-methyl oxime (ABP688) derivatives as metabotropic glutamate receptor subtype 5 PET radiotracers. Journal of Medicinal Chemistry, 55(16):7154-7162.

Gündüz, M; Şafak, C; Kaygısız, B; Koşar, B; Şimşek, R; Erol, K; Linden, Anthony (2012). Synthesis of Cyclopentapyridine and Thienopyridine derivatives as potential calcium channel modulators. Arzneimittelforschung, 62(4):167-175.

Mwinyi, Jessica; Grete-Wenger, Christa; Eloranta, Jyrki J; Kullak-Ublick, Gerd A (2012). The impact of PPARγ genetic variants on IBD susceptibility and IBD disease course. PPAR Research, 2012:349469.

Sirgel, Frederick A; Warren, Robin M; Streicher, Elizabeth M; Victor, Thomas C; van Helden, Paul D; Böttger, Erik C (2012). embB 306 Mutations as Molecular Indicators to Predict Ethambutol Susceptibility in Mycobacterium tuberculosis. Chemotherapy, 58(5):358-363.


Mlostoń, G; Pieczonka, A M; Kowalczyk, E; Linden, Anthony; Heimgartner, H (2011). Synthesis and selected reactions of hydrazides containing an imidazole moiety. Helvetica Chimica Acta, 94(10):1764-1777.

Yang, X; Fox, T; Berke, H (2011). Ammonia borane as a metal free reductant for ketones and aldehydes: a mechanistic study. Tetrahedron, 67(37):7121-7127.

Zhou, Y; Linden, Anthony; Heimgartner, H (2011). Reactions of Imidoyl Isoselenocyanates with Aromatic 2-Amino N-Heterocycles and 1-Methyl-1H-imidazole. Helvetica Chimica Acta, 94(9):1575-1585.

Deniz, G; Akdis, M (2011). NK cell subsets and their role in allergy. Expert Opinion on Biological Therapy, 11(7):833-841.

Ernst, K-H; Berke, H (2011). Optical activity and Alfred Werner's coordination chemistry. Chirality, 23(3):187-189.

Heimgartner, H; Linden, Anthony; Mekhael, M K G (2011). Reactions with 4-Hydroxy-2-methylbutananilides – unexpected formation of a cyclopropanecarboxamide. Helvetica Chimica Acta, 94(1):28-37.

Donsante, A; Yi, L; Zerfas, P M; Brinster, L R; Sullivan, P; Goldstein, D S; Prohaska, J; Centeno, J A; Rushing, E; Kaler, S G (2011). ATP7A gene addition to the choroid plexus results in long-term rescue of the lethal copper transport defect in a Menkes disease mouse model. Molecular Therapy, 19(12):2114-2123.

Staub, P O; Schiestl, F P; Leonti, M; Weckerle, C S (2011). Chemical analysis of incense smokes used in Shaxi, Southwest China: a novel methodological approach in ethnobotany. Journal of Ethnopharmacology, 138(1):212-218.

Münch, R C; Mühlebach, M D; Schaser, T; Kneissl, S; Jost, C; Plückthun, A; Cichutek, K; Buchholz, C J (2011). DARPins: an efficient targeting domain for lentiviral vectors. Molecular Therapy, 19(4):686-693.

Mann, A; Thakur, G; Shukla, V; Singh, A K; Khanduri, R; Naik, R; Jiang, Y; Kalra, N; Dwarakanath, B S; Langel, U; Ganguli, M (2011). Differences in DNA condensation and release by lysine and arginine homopeptides govern their DNA delivery efficiencies. Molecular Pharmaceutics, 5(8):1729-1741.

Glaus, E; Schmid, F; Da Costa, R; Berger, W; Neidhardt, J (2011). Gene therapeutic approach using mutation-adapted U1 snRNA to correct a RPGR splice defect in patient-derived cells. Molecular Therapy, 19(5):936-941.

Grez, M; Reichenbach, J; Schwäble, J; Seger, R; Dinauer, M C; Thrasher, A J (2011). Gene therapy of chronic granulomatous disease: the engraftment dilemma. Molecular Therapy, 19(1):28-35.

Mäe, M; Armulik, A; Betsholtz, C (2011). Getting to know the cast - cellular interactions and signaling at the neurovascular unit. Current Pharmaceutical Design, 17(26):2750-2754.

Flütsch, A; Schroeder, T; Grütter, M G; Patzke, Greta R (2011). HIV-1 protease inhibition potential of functionalized polyoxometalates. Bioorganic & Medicinal Chemistry Letters, 21(4):1162-1166.

Ogunshola, O O (2011). In vitro modeling of the blood-brain barrier: Simplicity versus complexity. Current Pharmaceutical Design, 17(26):2755-2761.

Deichmann, A; Brugman, M H; Bartholomae, C C; Schwarzwaelder, K; et al (2011). Insertion sites in engrafted cells cluster within a limited repertoire of genomic areas after gammaretroviral vector gene therapy. Molecular Therapy, 19(11):2031-2039.

Rogano, F; Stojnic, D; Linden, Anthony; Abou-Hadeed, K; Hansen, H J (2011). Introduction of adjacent oxygen-functionalities in Dimethyl Heptalenedicarboxylates. Helvetica Chimica Acta, 94(7):1194-1215.

Wächter, R; Brenneisen, R; Hamburger, M; Mennet, M; Schnelle, M; Worel, A M; Simões-Wüst, Ana Paula; von Mandach, U (2011). Leaf press juice from Bryophyllum pinnatum (Lamarck) Oken induces myometrial relaxation. Phytomedicine, 19(1):74-82.

Bradacs, G; Heilmann, J; Weckerle, C S (2011). Medicinal plant use in Vanuatu: a comparative ethnobotanical study of three islands. Journal of Ethnopharmacology, 137(1):434-448.

Grattagliano, I; Russmann, S; Diogo, C V; Bonfrate, L; Oliveira, P J; Wang, D Q H; Portincasa, P (2011). Mitochondria in chronic liver disease. Current Drug Targets, 12(6):879-893.

Schott, H; Goltz, D; Schott, T C; Jauch, C; Schwendener, R A (2011). N(4)-[Alkyl-(hydroxyphosphono)phosphonate]-cytidine-new drugs covalently linking antimetabolites (5-FdU, araU or AZT) with bone-targeting bisphosphonates (alendronate or pamidronate). Bioorganic & Medicinal Chemistry, 19(11):3520-3526.

Gasser, Gilles; Ott, Ingo; Metzler-Nolte, Nils (2011). Organometallic anticancer compounds. Journal of Medicinal Chemistry, 54(1):3-25.

Weckerle, C S; Cabras, S; Castellanos, M E; Leonti, M (2011). Quantitative methods in ethnobotany and ethnopharmacology: considering the overall flora-hypothesis testing for over- and underused plant families with the Bayesian approach. Journal of Ethnopharmacology, 137(1):837-843.

Fiaschetti, G; Grotzer, M A; Shalaby, T; Castelletti, D; Arcaro, A (2011). Quassinoids: From traditional drugs to new cancer therapeutics. Current Medicinal Chemistry, 18(3):316-328.

Fu, C; Linden, Anthony; Heimgartner, H (2011). Reaction of optically active Oxiranes with Thiofenchone and 1-Methylpyrrolidine-2-thione. Formation of 1,3-Oxathiolanes and Thiiranes. Helvetica Chimica Acta, 94(5):773-784.

Huang, D; Caflisch, A (2011). Small molecule binding to proteins: affinity and binding/unbinding dynamics from atomistic simulations. ChemMedChem, 6(9):1578-1580.

Templin, C; Kränkel, N; Lüscher, T F; Landmesser, U (2011). Stem cells in cardiovascular regeneration: from preservation of endogenous repair to future cardiovascular therapies. Current Pharmaceutical Design, 17(30):3280-3294.

Hostanska, K; Melzer, J; Amon, A; Saller, R (2011). Suppression of interleukin (IL)-8 and human beta defensin-2 secretion in LPS-and/or IL-1-Beta-stimulated airway epithelial A 549 cells by herbal formulation against respiratory infections (BNO 1030). Journal of Ethnopharmacology, 134(2):228-233.

Dannecker-Dörig, I; Linden, Anthony; Heimgartner, H (2011). Synthesis of Poly-Aib Oligopeptides and Aib-Containing Peptides via the 'Azirine/Oxazolone Method', and their crystal structures. Helvetica Chimica Acta, 94(6):993-1011.

Stieger, B; Beuers, U (2011). The canalicular bile salt export pump BSEP (ABCB11) as a potential therapeutic target. Current Drug Targets, 12(5):661-670.

Murphy, M; Huber, R; Esser, S; Riedner, B A; Massimini, M; Ferrarelli, F; Ghilardi, M F; Tononi, G (2011). The cortical topography of local sleep. Current Topics in Medicinal Chemistry, 11(19):2438-2446.

Tabatabai, G; Tonn, J C; Stupp, R; Weller, M (2011). The role of integrins in glioma biology and anti-glioma therapies. Current Pharmaceutical Design, 17(23):2402-2410.

Blenn, C; Wyrsch, P; Althaus, F R (2011). The ups and downs of tannins as inhibitors of poly(ADP-ribose)glycohydrolase. Molecules, 16(2):1854-1877.

Sudano, I; Roas, S; Noll, G (2011). Vascular abnormalities in essential hypertension. Current Pharmaceutical Design, 17(28):3039-3044.


Mawad, N; Ghorbani-Salman Pour, F; Linden, Anthony; Heimgartner, H (2010). Synthesis and Crystal Structure of 3,3,6,6-Tetramethylmorpholine-2,5-dione, and its 5-Monothio- and 2,5-Dithio-Derivatives. Helvetica Chimica Acta, 93(12):2326-2346.

Heimgartner, H; Linden, Anthony; Mlostoń, Grzegorz; Obijalska, E (2010). Synthesis of Three-, Five-, and Six-Membered Heterocycles Derived from New β-Amino-α-trifluoromethyl Alcohols. Helvetica Chimica Acta, 93(9):1725-1736.

Ushkov, A V; Kuznetsov, M A; Linden, Anthony; Heimgartner, H (2010). Tri- and Tetra-Substituted N-Phthalimidoaziridines in 1,3-Dipolar Cycloaddition Reactions. Helvetica Chimica Acta, 93(5):847-862.

Melkko, S; Mannocci, L; Dumelin, C E; Villa, A; Sommavilla, R; Zhang, Y; Grütter, M; Keller, N; Jermutus, L; Jackson, R H; Scheuermann, J; Neri, D (2010). Isolation of a small-molecule inhibitor of the antiapoptotic protein Bcl-xL from a DNA-encoded chemical library. ChemMedChem, 5(4):584-590.

Atanassov, P K; Linden, Anthony; Heimgartner, H (2010). Synthesis of 1,3-Selenazol-2(3H)-imines. Helvetica Chimica Acta, 93(3):395-404.

Jessen, Henning Jacob; Gademann, Karl (2010). 4-Hydroxy-2-pyridone alkaloids: Structures and synthetic approaches. Natural Product Reports, 27(8):1168.

Rajendran, L; Knölker, H J; Simons, K (2010). Subcellular targeting strategies for drug design and delivery. Nature Reviews. Drug Discovery, 9(1):29-42.

El Rayes, S; Linden, Anthony; Abou-Hadeed, K; Hansen, H J (2010). Alkylation reactions at the benzo moiety of 2,4-Dimethoxy-3-(phenylsulfonyl)benzo[a]heptalenes – model compounds of colchicinoids. Helvetica Chimica Acta, 93(10):1894-1911.

Meyer, S; Vogt, T; Landthaler, M; Berand, A; Reichle, A; Bataille, F; Marx, A H; Menz, A; Hartmann, A; Kunz-Schughart, L A; Wild, P J (2010). Cyclooxygenase 2 (COX2) and peroxisome proliferator-activated receptor gamma (PPARG) are stage-dependent prognostic markers of malignant melanoma. PPAR research, 2010:848645.

Pistoia, F; Cipollone, F; Ferri, C; Sarà, M; Sudano, I; Desideri, G B (2010). Cyclooxygenase and atherosclerosis: a smoking area. Current Pharmaceutical Design, 16(23):2567-2571.

Jin, X; Linden, Anthony; Hansen, H J (2010). Formation of 6-Methyl-7,11-diphenylheptaleno[1,2-c]furanones. Helvetica Chimica Acta, 93(5):934-945.

Jung, H H; Bremer, J; Weller, M (2010). Gene therapy for myositis. In: Chernajovsky, Y; Robbins, P D. Gene therapy for autoimmune and inflammatory. Basel: Birkhäuser, 79-90.

Besler, C; Heinrich, K; Riwanto, M; Lüscher, T F; Landmesser, U (2010). High-density lipoprotein-mediated anti-atherosclerotic and endothelial-protective effects: a potential novel therapeutic target in cardiovascular disease. Current Pharmaceutical Design, 16(13):1480-1493.

Zhou, T; Caflisch, A (2010). High-throughput virtual screening using quantum mechanical probes: discovery of selective kinase inhibitors. ChemMedChem, 5(7):1007-1014.

Simões-Wüst, Ana Paula; Grãos, M; Duarte, C B; Brenneisen, R; Hamburger, M; Mennet, M; Ramos, M H; Schnelle, M; Wächter, R; Worel, A M; von Mandach, U (2010). Juice of Bryophyllum pinnatum (Lam.) inhibits oxytocin-induced increase of the intracellular calcium concentration in human myometrial cells. Phytomedicine, 17(12):980-6.

Mindt, Thomas L; Struthers, Harriet; Spingler, Bernhard; Brans, Luc; Tourwe, Dirk; Garcia-Garayoa, Elisa; Schibli, Roger (2010). Molecular assembly of multifunctional Tc-99m radiopharmaceuticals using "clickable" amino acid derivatives. ChemMedChem, 5(12):2026-2038.

Gademann, K; Portmann, C; Blom, J F; Zeder, M; Jüttner, F (2010). Multiple toxin production in the cyanobacterium microcystis: isolation of the toxic protease inhibitor cyanopeptolin 1020. Journal of Natural Products, 73(5):980-984.

Dummer, R; Eichmüller, S; Gellrich, S; Assaf, C; Dreno, B; Schiller, M; Dereure, O; Baudard, M; Bagot, M; Khammari, A; Bleuzen, P; Bataille, V; Derbij, A; Wiedemann, N; Waterboer, T; Lusky, M; Acres, B; Urosevic-Maiwald, M (2010). Phase II clinical trial of intratumoral application of TG1042 (adenovirus-interferon-gamma) in patients with advanced cutaneous T-cell lymphomas and multilesional cutaneous B-cell lymphomas. Molecular Therapy, 18(6):1244-1247.

Aguzzi, A; O'Connor, T (2010). Protein aggregation diseases: pathogenicity and therapeutic perspectives. Nature Reviews. Drug Discovery, 9(3):237-248.

Zhou, T; Huang, D; Caflisch, A (2010). Quantum mechanical methods for drug design. Current Topics in Medicinal Chemistry, 10(1):33-45.

Michalakis, Stylianos; Mühlfriedel, Regine; Tanimoto, Naoyuki; Krishnamoorthy, Vidhyasankar; Koch, Susanne; Fischer, M Dominik; Becirovic, Elvir; Bai, Lin; Huber, Gesine; Beck, Susanne C; Fahl, Edda; Büning, Hildegard; Paquet-Durand, François; Zong, Xiangang; Gollisch, Tim; Biel, Martin; Seeliger, Mathias W (2010). Restoration of Cone Vision in the CNGA3$^{−/−}$ Mouse Model of Congenital Complete Lack of Cone Photoreceptor Function. Molecular Therapy, 18(12):2057-2063.

Kindermann, M; Roschitzki-Voser, H; Caglic, D; Repnik, U; Miniejew, C; Mittl, P R E; Kosec, G; Grütter, M G; Turk, B; Wendt, K U (2010). Selective and sensitive monitoring of caspase-1 activity by a novel bioluminescent activity-based probe. Chemistry & Biology, 17(9):999-1007.

Zonta, C; De Lucchi, O; Linden, Anthony; Lutz, M (2010). Synthesis and structure of D3h-symmetric triptycene trimaleimide. Molecules, 15(1):226-232.

Jin, X; Linden, Anthony; Hansen, H J (2010). Synthesis of 1-methyl-6,10-diphenylheptalene derivatives. Helvetica Chimica Acta, 93(4):729-745.

Leonti, M; Cabras, S; Weckerle, C S; Solinas, M N; Casu, L (2010). The causal dependence of present plant knowledge on herbals: contemporary medicinal plant use in Campania (Italy) compared to Matthioli (1568). Journal of Ethnopharmacology, 130(2):379-391.

Abela, I A; Reynell, L; Trkola, A (2010). Therapeutic antibodies in HIV treatment - classical approaches to novel advances. Current Pharmaceutical Design, 16(33):3754-3766.

Veit, O; Hatz, C; Niedrig, M; Furrer, H J (2010). Yellow fever vaccination in HIV-infected patients. HIV Therapy, 4(1):17-26.


Jacob, F; Goldstein, D R; Fink, D; Heinzelmann-Schwarz, V (2009). Proteogenomic studies in epithelial ovarian cancer: established knowledge and future needs. Biomarkers in Medicine, 3(6):743-756.

Mlostoń, Grzegorz; Urbaniak, K; Domagała, M; Pfitzner, A; Zabel, M; Heimgartner, H (2009). Thermal [2+3]-cycloadditions of trans-1-methyl-2,3-diphenylaziridine with C=S and C=C dipolarophiles: An unexpected course with dimethyl dicyanofumarate. Helvetica Chimica Acta, 92(12):2631-2642.

Wenger, R H; Camenisch, G; Stiehl, D P; Katschinski, D M (2009). HIF Prolyl-4-hydroxylase Interacting Proteins: Consequences for Drug Targeting. Current Pharmaceutical Design, 15(33):3886-3894.

Mlostoń, Grzegorz; Urbaniak, K; Linden, Anthony; Heimgartner, H (2009). A new approach to 2,2-disubstituted 1-(methylsulfanyl)vinyl phosphonates via an intermediate thiocarbonyl ylide. Tetrahedron, 65(39):8191-8198.

Seyfried, M S; Linden, Anthony; Mlostoń, Grzegorz; Heimgartner, H (2009). Chemoselectivity of the Reactions of Diazomethanes with 5-Benzylidene-3-phenylrhodanine. Helvetica Chimica Acta, 92(9):1800-1816.

Mlostoń, Grzegorz; Celeda, M; Linden, Anthony; Heimgartner, H (2009). Two- and Three-Component Reactions Leading to New Enamines Derived from 2,3-Dicyanobut-2-enoates. Helvetica Chimica Acta, 92(8):1520-1537.

Weckerle, C S; Ineichen, R; Huber, F K; Yang, Y (2009). Mao's heritage: medicinal plant knowledge among the Bai in Shaxi, China, at a crossroad between distinct local and common widespread practice. Journal of Ethnopharmacology, 123(2):213-228.

Bülbül, B; Öztürk, G S; Vural, M; Simsek, R; Sarioglu, Y; Linden, Anthony; Ülgen, M; Safak, C (2009). Condensed 1,4-dihydropyridines with various esters and their calcium channel antagonist activities. European Journal of Medicinal Chemistry, 44(5):2052-2058.

Zeilhofer, Hanns Ulrich; Witschi, R; Hösl, K (2009). Subtype-selective GABA(A) receptor mimetics-novel antihyperalgesic agents? Journal of Molecular Medicine, 87(5):465-469.

Zou, C; Kumaran, S; Walser, R; Zerbe, O (2009). Properties of the N-terminal domains from Y receptors probed by NMR spectroscopy. Journal of Peptide Science, 15(3):184-191.

Linden, Anthony; Petridis, A; James, B D (2009). Structural Diversity in Thallium Chemistry. Part VI. Analysis of Structure Correlation in Organoammonium Bromothallates(III). Helvetica Chimica Acta, 92(1):29-71.

Schott, H; Hamprecht, K; Schott, S; Schott, T C; Schwendener, R (2009). Synthesis and in vitro activities of a new antiviral duplex drug linking Zidovudine (AZT) and Foscarnet (PFA) via an octadecylglycerol residue. Bioorganic & Medicinal Chemistry, 17(1):303-310.

Mindt, T L; Schweinsberg, C; Brans, L; Hagenbach, A; Abram, U; Tourwé, D; Garcia-Garayoa, E; Schibli, R (2009). A click approach to structurally diverse conjugates containing a central di-1,2,3-triazole metal chelate. ChemMedChem, 4(4):529-539.

Uehleke, B; Stange, R (2009). A clinical surrogate model for proof of efficacy of external phytomedicines for muscle pain. Results of a randomized, placebo-controlled clinical study in volunteers with muscle pain due to physical training. Phytomedicine, 16(6-7):509-512.

Iten, F; Saller, R; Abel, G; Reichling, J (2009). Additive antimicrobial [corrected] effects of the active components of the essential oil of Thymus vulgaris--chemotype carvacrol. Planta Medica, 75(11):1231-1236.

Russmann, S; Kullak-Ublick, G A; Grattagliano, I (2009). Current concepts of mechanisms in drug-induced hepatotoxicity. Current Medicinal Chemistry, 16(23):3041-3053.

Friedman, R; Caflisch, A (2009). Discovery of plasmepsin inhibitors by fragment-based docking and consensus scoring. ChemMedChem, 4(8):1317-1326.

Rickenbacher, A; Breitenstein, S; Lesurtel, M; Frilling, A (2009). Efficacy of TachoSil a fibrin-based haemostat in different fields of surgery - a systematic review. Expert Opinion on Biological Therapy, 9(7):897-907.

Ekonomiuk, D; Su, X C; Ozawa, K; Bodenreider, C; Lim, S P; Otting, G; Huang, D; Caflisch, A (2009). Flaviviral protease inhibitors identified by fragment-based library docking into a structure generated by molecular dynamics. Journal of Medicinal Chemistry, 52(15):4860-4868.

Blank, P R; Szucs, T D (2009). Increasing influenza vaccination coverage in recommended population groups in Europe. Expert Review of Vaccines, 8(4):425-433.

Dumitru, C A; Sandalcioglu, I E; Wagner, M; Weller, M; Gulbins, E (2009). Lysosomal ceramide mediates gemcitabine-induced death of glioma cells. Journal of Molecular Medicine, 87(11):1123-1132.

Bonmarin, M; Helbing, J (2009). Polarization control of ultrashort mid-IR laser pulses for transient vibrational circular dichroism measurements. Chirality, 21(1E):E298-E306.

Obrecht, D; Robinson, J A; Bernardini, F; Bisang, C; DeMarco, S J; Moehle, K; Gombert, F O (2009). Recent progress in the discovery of macrocyclic compounds as potential anti-infective therapeutics. Current Medicinal Chemistry, 16(1):42-65.

Lafleur, K; Huang, D; Zhou, T; Caflisch, A; Nevado, C (2009). Structure-based optimization of potent and selective inhibitors of the tyrosine kinase erythropoietin producing human hepatocellular carcinoma receptor B4 (EphB4). Journal of Medicinal Chemistry, 52(20):6433-6446.

Collin, M P; Hobbie, S N; Böttger, E C; Vasella, A (2009). Synthesis and Evaluation of S- and C(1)-Substituted Analogues of Lincomycin. Helvetica Chimica Acta, 92(2):230-266.

Schott, H; Schott, S; Schwendener, R (2009). Synthesis and in vitro activities of new anticancer duplex drugs linking 2'-deoxy-5-fluorouridine (5-FdU) with 3'-C-ethynylcytidine (ECyd) via a phosphodiester bonding. Bioorganic & Medicinal Chemistry, 17(19):6824-6831.

Ebbesen, P; Pettersen, E O; Gorr, T A; Jobst, G; Williams, K; Kieninger, J; Wenger, R H; Pastorekova, S; Dubois, L; Lambin, P; Wouters, B G; Van den Beucken, T; Supuran, C T; Poellinger, L; Ratcliffe, P; Kanopka, A; Görlach, Agnes; Gassmann, Max; Harris, A L; Maxwell, P; Scozzafava, A (2009). Taking advantage of tumor cell adaptations to hypoxia for developing new tumor markers and treatment strategies. Journal of Enzyme Inhibition and Medicinal Chemistry, 24(S1):1-39.

Grotzer, M A; Castelletti, D; Fiaschetti, G; Shalaby, T; Arcaro, A (2009). Targeting Myc in pediatric malignancies of the central and peripheral nervous system. Current Cancer Drug Targets, 9(2):176-188.

Scocchi, M; Lüthy, C; Decarli, P; Mignogna, G; Christen, P; Gennaro, R (2009). The proline-rich antibacterial peptide Bac7 binds to and inhibits in vitro the molecular chaperone DnaK. International Journal of Peptide Research and Therapeutics, 15(2):147-155.

Akdis, M; Akdis, C A (2009). Therapeutic manipulation of immune tolerance in allergic disease. Nature Reviews. Drug Discovery, 8(8):645-660.

Bolliger, J L; Frech, C M (2009). Transition metal-free amination of aryl halides-A simple and reliable method for the efficient and high-yielding synthesis of N-arylated amines. Tetrahedron, 65(6):1180-1187.


von Eckardstein, A (2008). HDL - a difficult friend. Drug Discovery Today, 5(3-4):e315-e324.

Landolt, H P (2008). Genotype-dependent differences in sleep, vigilance and response to stimulants. Current Pharmaceutical Design, 14(32):3396-3407.

Christiansen, G; Yoshida, W Y; Blom, J F; Portmann, C; Gademann, K; Hemscheidt, T; Kurmayer, R (2008). Isolation and structure determination of two microcystins and sequence comparison of the McyABC aenylation domains in Planktothrix species. Journal of Natural Products, 71(11):1881-1886.

Jeremic, T; Linden, Anthony; Heimgartner, H (2008). New 21- and 24-atom Aib-containing cyclopeptides. Journal of Peptide Science, 14(9):1051-1061.

Malashikhin, S A; Linden, Anthony; Heimgartner, H; Rodina, L L; Nikolaev, V A (2008). Synthesis and structures of two isomeric 4-diazo-2,3,4,5-tetrahydrofuran-3-ones. Helvetica Chimica Acta, 91(9):1662-1668.

Seeger, M A; Diederichs, K; Eicher, T; Brandstätter, L; Schiefner, A; Verrey, F; Pos, K M (2008). The AcrB efflux pump: conformational cycling and peristalsis lead to multidrug resistance. Current Drug Targets, 9(9):729-749.

Pathak, Rashmi; Perez-Fernandez, Déborah; Nandurdikar, Rahul; Kalapala, Sarath K; Böttger, Erik C; Vasella, Andrea (2008). Synthesis and evaluation of paromomycin derivates modified at C(4'). Helvetica Chimica Acta, 91(8):1533-1552.

Mlostoń, Grzegorz; Woźnicka, M; Drabowicz, J; Linden, Anthony; Heimgartner, H (2008). Addition reactions of sulfenyl and sulfinyl chlorides with 3-phenyl-1-azabicyclo[1.1.0]butane. Helvetica Chimica Acta, 91(8):1419-1429.

Bisegger, P; Manov, N; Bienz, S (2008). Solid-phase synthesis of cyclic polyamines. Tetrahedron, 64(32):7531-7536.

Marti, F; Steffen, Robert; Mütsch, Margot (2008). Influenza vaccine: a travelers’ vaccine? Expert Review of Vaccines, 7(5):679-687.

Amoroso, A; Crespan, E; Wimmer, U; Hubscher, U; Maga, G (2008). DNA Polymerases and Oxidative Damage: Friends or Foes? Current Molecular Pharmacology, 1(2):162-170.

Hausmann, M; Rogler, G (2008). Immune-non immune networks in intestinal inflammation. Current Drug Targets, 9(5):388-394.

Dummer, R; Rochlitz, C; Velu, T; Acres, B; Limacher, J M; Bleuzen, P; Lacoste, G; Slos, P; Romero, P; Urosevic, M (2008). Intralesional adenovirus-mediated interleukin-2 gene transfer for advanced solid cancers and melanoma. Molecular Therapy, 16(5):985-994.

Belousova, E A; Crespan, E; Lebedeva, N A; Rechunova, N J; Hübscher, U; Maga, G; Lavrik, O I (2008). Photoreactive DNA Probes as a Tool for Studying the Translesion Synthesis System in Mammalian Cell Extracts. Medicinal Chemistry, 4(2):155-162.

Lorenzi, I; von Eckardstein, A; Cavelier, C; Radosavljevic, S; Rohrer, L (2008). Apolipoprotein A-I but not high-density lipoproteins are internalised by RAW macrophages: roles of ATP-binding cassette transporter A1 and scavenger receptor BI. Journal of Molecular Medicine, 86(2):171-183.

Sommen, G L; Linden, Anthony; Heimgartner, H (2008). Selenium-containing heterocycles from isoselenocyanates:5-methylselenazole derivatives from the reaction with malononitrile and propargyl chloride. Helvetica Chimica Acta, 91(2):209-219.

Cortes, M L; Oehmig, A; Saydam, O; Sanford, J D; Perry, K F; Fraefel, C; Breakefield, X (2008). Targeted integration of functional human ATM cDNA into genome mediated by HSV/AAV hybrid amplicon vector. Molecular Therapy, 16(1):81-88.

Landmesser, T; Linden, Anthony; Hansen, H J (2008). A novel route to 1-substituted 3-(dialkylamino)-9-oxo-9H-indeno[2,1-c]pyridine-4-carbonitriles. Helvetica Chimica Acta, 91(2):265-284.

Wolf, S A; Tauber, S; Ullrich, O (2008). CNS immune surveillance and neuroinflammation: endocannabinoids keep control. Current Pharmaceutical Design, 14(23):2266-2278.

Bauer, V L; Braselmann, H; Henke, M; Mattern, D; Walch, A; Unger, K; Baudis, Michael; Lassmann, S; Huber, R; Wienberg, J; Werner, M; Zitzelsberger, H F (2008). Chromosomal changes characterize head and neck cancer with poor prognosis. Journal of Molecular Medicine, 86(12):1353-1365.

Ding, Z; Harding, C O; Rebuffat, A; Elzaouk, L; Wolff, J A; Thöny, B (2008). Correction of murine PKU following AAV-mediated intramuscular expression of a complete phenylalanine hydroxylating system. Molecular Therapy, 16(4):673-681.

Kolb, P; Huang, D; Dey, F; Caflisch, A (2008). Discovery of kinase inhibitors by high-throughput docking and scoring based on a transferable linear interaction energy model. Journal of Medicinal Chemistry, 51(5):1179-1188.

Hippert, C; Dubois, G; Morin, C; Disson, O; Ibanes, S; Jacquet, C; Schwendener, R; Antignac, C; Kremer, E J; Kalatzis, V (2008). Gene transfer may be preventive but not curative for a lysosomal transport disorder. Molecular Therapy, 16(8):1372-1381.

Zhou, T; Huang, D; Caflisch, A (2008). Is quantum mechanics necessary for predicting binding free energy? Journal of medicinal chemistry, 51(14):4280-4288.

Rudin, M (2008). Noninvasive imaging of receptor function: signal transduction pathways and physiological readouts. Current Opinion in Drug Discovery and Development, 11(5):606-615.

Mann, A; Thakur, G; Shukla, V; Ganguli, M (2008). Peptides in DNA delivery: current insights and future directions. Drug Discovery Today, 13(3-4):152-160.

Neglia, D; Rimoldi, O; Kaufmann, P A; Camici, P G (2008). Radionuclide PET and PET/CT in coronary artery disease. Current Pharmaceutical Design, 14(18):1798-814.

Brun, K A; Linden, Anthony; Heimgartner, H (2008). Synthesis and conformational analysis of pentapeptides containing enantiomerically pure 2,2-disubstituted glycines. Helvetica Chimica Acta, 91(3):526-558.

Jasiński, M; Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, H (2008). Synthesis and selected transformations of 1H-imidazole 3-oxides derived from amino acid esters. Helvetica Chimica Acta, 91(10):1916-1933.

Collin, M P; Hobbie, S N; Böttger, E C; Vasella, A (2008). Synthesis of 1,2,3-triazole analogues of lincomycin. Helvetica Chimica Acta, 91(10):1838-1848.

Mlostoń, Grzegorz; Mucha, P; Urbaniak, K; Broda, K; Heimgartner, H (2008). Synthesis of optically active 1-(1-phenylethyl)imidazoles eerived from 1-phenylethylamine. Helvetica Chimica Acta, 91(2):232-238.

Akdis, M (2008). T-cell tolerance to inhaled allergens: mechanisms and therapeutic approaches. Expert Opinion on Biological Therapy, 8(6):769-777.

Budzowski, A; Linden, Anthony; Heimgartner, H (2008). The azirine/oxazolone approach to the synthesis of Aib-Pro endothiopeptides. Helvetica Chimica Acta, 91(8):1471-1488.


Knipp, M; Karotki, A V; Chesnov, S; Natile, G; Sadler, P J; Brabec, V; Vasák, M (2007). Reaction of Zn7metallothionein with cis- and trans-[Pt(N-donor)2Cl2] anticancer complexes: trans-Pt(II) complexes retain their N-donor ligands. Journal of Medicinal Chemistry, 50(17):4075-4086.

Döbbeling, U (2007). Transcription factor profiling shows new ways towards new treatment options of cutaneous T cell lymphomas. Current Drug Discovery Technologies, 4(1):24-30.

Egli, D H; Linden, Anthony; Heimgartner, H (2007). 1,5-Dipolar electrocyclizations of Thiocarbonyl Ylides bearing C=N groups: Reactions of N-[(Dimethylamino)methylene]thiobenzamide and 2-(Dimethylhydrazono)-1-phenylethane-1-thione with Diazo compounds. Helvetica Chimica Acta, 90(1):86-100.

Mlostoń, Grzegorz; Woźnicka, M; Heimgartner, H (2007). 5-Morpholino-1,2,3,4-thiatriazole as a Sulfur-Transfer reagent in the reactions with Thioketones. Helvetica Chimica Acta, 90(3):594-600.

Battegay, E; Demiguel, L; Petrimpol, M; Humar, R (2007). Effects of anti-hypertensive drugs on vessel rarefactio. Current Opinion in Pharmacology, 7(2):151-157.

Gerber, U; Gee, C E; Benquet, P (2007). Metabotropic glutamate receptors: intracellular signaling pathways. Current Opinion in Pharmacology, 7(1):56-61.

Mlostoń, Grzegorz; Warkentin, J; Linden, Anthony; Heimgartner, H (2007). Reactions of dimethoxycarbene with N-tosylated imines. Helvetica Chimica Acta, 90(10):2024-2036.

Romański, J; Mlostoń, Grzegorz; Heimgartner, H (2007). Reactions of polycyclic ketones with Dimethoxycarbene; a convenient route for a one-pot preparation of some alpha-hydroxycarboxylic acid esters. Helvetica Chimica Acta, 90(7):1279-1288.

Sommen, G L; Linden, Anthony; Heimgartner, H (2007). Selenium-Containing heterocycles from isoselenocyanates: synthesis of 5-Amino-2,4-dihydro-3H-1,2,4-triazole-3-selones. Helvetica Chimica Acta, 90(4):641-651.

Sommen, G L; Linden, Anthony; Heimgartner, H (2007). Selenium-containing heterocycles from Isoselenocyanates: Synthesis of 1,3-Selenazinane and 1,3-Selenazinanone derivatives. Helvetica Chimica Acta, 90(3):472-487.

Sommen, G L; Linden, Anthony; Heimgartner, H (2007). Selenium-containing heterocycles from isoselenocyanates: Base-catalyzed reaction of malononitrile with phenyl isoselenocyanate and bromoacetonitrile or alpha-halogenated ketones. Helvetica Chimica Acta, 90(10):1849-1855.

Jasiński, M; Mlostoń, Grzegorz; Mucha, P; Linden, Anthony; Heimgartner, H (2007). Synthesis of new Bis-imidazole derivatives. Helvetica Chimica Acta, 90(9):1765-1780.

Mlostoń, Grzegorz; Heimgartner, H (2007). The first reaction of Dimethoxycarbene with an imine moiety. Helvetica Chimica Acta, 90(9):1758-1764.

Nikolaev, V V; Linden, Anthony; Heimgartner, H (2007). Thermolysis of imidates: A new method for the generation of carbonyl ylides. Helvetica Chimica Acta, 90(12):2330-2341.


Nett, P C; Teixeira, M M; Candinas, D; Barton, M (2006). Recent developments on endothelin antagonists as immunomodulatory drugs - from infection to transplantation medicine. Recent Patents on Cardiovascular Drug Discovery, 1(3):265-276.

Sobek, J; Bartscherer, K; Jacob, A; Hoheisel, J D; Angenendt, P (2006). Microarray technology as a universal tool for high-throughput analysis of biological systems. Combinatorial chemistry & high throughput screening, 9(5):365-380.

Egli, D H; Linden, Anthony; Heimgartner, H (2006). 1,5-Dipolar electrocyclizations in reactions of alpha-Thioxo Ketones and alpha-Thioxo Thioamides with Diazo compounds. Helvetica Chimica Acta, 89(9):1910-1926.

Iliev, Boyan; Linden, Anthony; Kunz, Roland; Heimgartner, Heinz (2006). 14-Membered cyclodepsipeptides with alternating beta-hydroxy and alpha-amino acids by cyclodimerization. Tetrahedron, 62(6):1079-1094.

Nikolaev, Vsevolod; Hennig, Lothar; Heimgartner, Heinz; Schulze, Bärbel; Nikolaev, Valerij (2006). Dual reactivity of imidic carbonyl ylides in Rh(II)-catalyzed reactions of alpha-diazocarbonyl compounds with succinimide. Tetrahedron Letters, 47(15):2643-2647.

Stamm, S; Heimgartner, H (2006). Introduction of the Aib-Pro unit into peptides by means of the ‘azirine/oxazolone method’ on solid phase. Tetrahedron, 62(41):9671-9680.

Stamm, S; Heimgartner, H (2006). Novel N-(2,2-Dimethyl-2H-azirin-3-yl)-L-prolinates as Aib-Pro Synthons. Helvetica Chimica Acta, 89(9):1841-1855.

Lesniak, S; Mloston, G; Urbaniak, K; Wasiak, P; Linden, Anthony; Heimgartner, H (2006). Phosphonylated thiocarbonyl ylides from the reaction of aromatic thioketones with diethyl diazomethylphosphonates. Tetrahedron, 62(33):7776-7782.

Iliev, Boyan; Linden, Anthony; Heimgartner, Heinz (2006). Reaction of gamma-Hydroxy-N-[1-(dimethylcarbamoyl)ethyl]butanamides under the ‘Direct Amide Cyclization’ Conditions. Helvetica Chimica Acta, 89(1):153-175.

Mlostoń, Grzegorz; Jasiński, M; Linden, Anthony; Heimgartner, H (2006). Reactions of 2-unsubstituted 1H-Imidazole 3-Oxides with 2,2- Bis(trifluoromethyl)ethene-1,1-dicarbonitrile: A stepwise 1,3-dipolar Cycloaddition. Helvetica Chimica Acta, 89(7):1304-1316.

Majchrzak, A; Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, H (2006). Reactions of Chlorosulfanyl Derivatives of Cyclobutanones with Different Nucleophiles. Helvetica Chimica Acta, 89(5):1042-1061.

Egli, D H; Linden, Anthony; Heimgartner, H (2006). Reactions of Thioketones possessing a conjugated C=C bond with Diazo compounds. Helvetica Chimica Acta, 89(12):3041-3055.

Egli, D H; Linden, Anthony; Heimgartner, H (2006). Reactions of alpha,beta-unsaturated Thioamides with Diazo compounds. Helvetica Chimica Acta, 89(11):2815-2824.

Fedorov, A; Fu, C; Heimgartner, H (2006). Regio- and stereoselectivity in the Lewis acid- and NaH-induced reactions of thiocamphor with (R)-2-vinyloxirane. Helvetica Chimica Acta, 89(3):456-467.

Sommen, G L; Linden, Anthony; Heimgartner, H (2006). Selenium-containing Heterocycles from Isoselenocyanates: Use of Hydrazine for the synthesis of 1,3,4-Selenadiazine derivatives. Helvetica Chimica Acta, 89(7):1322-1329.

Sommen, G L; Linden, Anthony; Heimgartner, H (2006). Selenium-containing heterocycles from isoselenocyanates: synthesis of 2-methylidene-1,3-selenazolidine derivatives. Tetrahedron, 62:3344-3354.

Köttgen, P; Linden, Anthony; Heimgartner, H (2006). Synthesis of Enniatin-like Cyclic Depsipeptides via direct Amide Cyclization. Helvetica Chimica Acta, 89(4):731-746.

Mlostoń, Grzegorz; Heimgartner, H (2006). The first ring-enlargement of a 1-Azabicyclo[1.1.0]butane to a 1-Azabicyclo[2.1.1]hexane. Helvetica Chimica Acta, 89(3):442-449.

Stamm, Simon; Linden, Anthony; Heimgartner, Heinz (2006). The ‘Azirine/Oxazolone Method’ on solid phase: Introduction of various alpha,alpha-disubstituted alpha-Amino Acids. Helvetica Chimica Acta, 89(1):1-15.

Iliev, Boyan; Verma, Sanjiv; Linden, Anthony; Heimgartner, Heinz (2006). Transformation of 5-Hydroxy- to (5-Chloropentanoyl)amino Derivatives under ‘Direct Amide Cyclization’ Conditions. Helvetica Chimica Acta, 89(2):352-359.


Shakhova, Olga; Leung, Carly; Marino, Silvia (2005). Bmi1 in development and tumorigenesis of the central nervous system. Journal of Molecular Medicine, 83(8):596-600.

Buterin, T; Meyer, C; Giese, B; Naegeli, H (2005). DNA quality control by conformational readout on the undamaged strand of the double helix. Chemistry & Biology, 12(8):913-922.

Bienz, Stefan; Bisegger, Pascal; Guggisberg, Armin; Hesse, Manfred (2005). Polyamine alkaloids. Natural Product Reports, 22(5):647-658.

Brun, Kathrin A; Heimgartner, Heinz (2005). A new 2H-Azirin-3-amine as a synthon for 2-Methylaspartate. Helvetica Chimica Acta, 88(11):2951-2959.

Philipova, Irena; Linden, Anthony; Heimgartner, Heinz (2005). Application of the "Direct Amide Cyclization" to Peptides Containing an Anthranilic Acid Residue. Helvetica Chimica Acta, 88:1711-1733.

Sommen, Geoffroy L; Linden, Anthony; Heimgartner, Heinz (2005). First synthesis of a selenazepane. Tetrahedron Letters, 46(39):6723-6725.

Robinson, J A; Shankaramma, S C; Jetter, P; Kienzl, U; Schwendener, R; Vrijbloed, J W; Obrecht, D (2005). Properties and structure-activity studies of cyclic beta-hairpin peptidomimetics based on the cationic antimicrobial peptide protegrin I. Bioorganic & Medicinal Chemistry, 13(6):2055-2064.

Malaschichin, Sergej; Fu, Changchun; Linden, Anthony; Heimgartner, Heinz (2005). Ring enlargement and sulfur-transfer processes in SiO2-catalyzed reactions of thiocarbonyl compounds with optically active oxiranes. Helvetica Chimica Acta, 88(12):3253-3262.

Sommen, Geoffroy L; Linden, Anthony; Heimgartner, Heinz (2005). Selenium-Containing Heterocycles from Isoselenocyanates: Cycloaddition of Carbodiimides to Selenazetidines. Helvetica Chimica Acta, 88(4):766-773.

Ludwig, P S; Schwendener, R; Schott, H (2005). Synthesis and anticancer activities of amphiphilic 5-fluoro-2'-deoxyuridylic acid prodrugs. European Journal of Medicinal Chemistry, 40(5):494-504.

Jeremic, Tatjana; Linden, Anthony; Möhle, Kerstin; Heimgartner, Heinz (2005). Synthesis and conformational analysis of 18-membered Aib-containing cyclohexapeptides. Tetrahedron, 61(7):1871-1883.

Mlostoń, Grzegorz; Majchrzak, Agnieszka; Rutkowska, Marzena; Woznicka, Marta; Linden, Anthony; Heimgartner, Heinz (2005). Synthesis and reactions of a new cyclobutanethione derivative. Helvetica Chimica Acta, 88(10):2624-2636.

Mlostoń, Grzegorz; Urbaniak, Katarzyna; Gulea, Mihaela; Masson, Serge; Linden, Anthony; Heimgartner, Heinz (2005). [2+3]-Cycloadditions of Phosphonodithioformate S-Methanides with C=S, N=N, and C=C Dipolarophiles. Helvetica Chimica Acta, 88(10):2582-2592.


Manov, Nikolay; Tzouros, Manuel; Bigler, Laurent; Bienz, Stefan (2004). Solid-phase synthesis of 15N-labeled acylpentamines as reference compounds for the MS/MS investigation of spider toxins. Tetrahedron, 60(10):2387-2391.

Meier, O; Greber, U F (2004). Adenovirus endocytosis. Journal of Gene Medicine, 6(S1):S152-S163.

Hilty, Florentine M; Brun, Kathrin A; Heimgartner, Heinz (2004). A New 2H-Azirin-3-amine as a Synthon for α-Methyl Glutamate. Helvetica Chimica Acta, 87(10):2539-2548.

Schiltz, J G; Salzer, U; Mohajeri, M H; Franke, D; Heinrich, J; Pavlovic, J; Wollmer, M A; Nitsch, R M; Moelling, K (2004). Antibodies from a DNA peptide vaccination decrease the brain amyloid burden in a mouse model of Alzheimer's disease. Journal of Molecular Medicine, 82(10):706-714.

Mekhael, Maged K G; Bienz, Stefan; Linden, Anthony; Heimgartner, Heinz (2004). Azirine/Oxindole ring enlargement via Amidinium intermediates. Helvetica Chimica Acta, 87(9):2385-2404.

Atanassov, Plaen K; Linden, Anthony; Heimgartner, Heinz (2004). Derivatives from Isoselenocyanates: Synthesis of 2-Phenyl-6H-[5,1,3]benzoselenadiazocine. Helvetica Chimica Acta, 87:1452-1466.

Bienz, Stefan; Hesse, Manfred (2004). Eine neue Synthese von Muscon undExalton®: Die Enamin-Route der Ringerweiterungsreaktion. Helvetica Chimica Acta, 71(7):1704-1707.

Fässler, Jürg; Huber, Priska; Bratovanov, Svetoslav; Bigler, Laurent; Bild, Norbert; Bienz, Stefan (2004). Neighboring-Group participation in the gas phase. Loss of benzaldehyde from [(benzyloxy)methyl]dialkylsilyl-substituted 1,3-dithianes. Helvetica Chimica Acta, 78(7):1855-1862.

Urbaniak, Katarzyna; Szymański, Radoslaw; Romański, Jaroslaw; Mlostoń, Grzegorz; Domagala, Malgorzata; Linden, Anthony; Heimgartner, Heinz (2004). New Studies on [2 + 3] Cycloadditions of Thermally Generated N-Isopropyl- and N-(4-Methoxyphenyl)-Substituted Azomethine Ylides. Helvetica Chimica Acta, 87:496-510.

Chen, F; David, D; Ferrari, A; Götz, J (2004). Posttranslational modifications of tau - role in human tauopathies and modeling in transgenic animals. Current Drug Targets, 5(6):503-515.

Majchrzak, Agnieszka; Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (2004). Reactions of Sulfanyl Chlorides with Thiocamphor and Thiofenchone: Wagner-Meerwein Rearrangement of an Intermediate Thiocarbonylium Ion. Helvetica Chimica Acta, 87:790-799.

Fu, Changchun; Linden, Anthony; Heimgartner, Heinz (2004). Regio- and stereoselective 1,3-Oxathiolane formation in the reaction of Thiolactones with optically active oxiranes. Helvetica Chimica Acta, 87(9):2296-2309.

Fu, Changchun; Thrane, Marie V; Linden, Anthony; Heimgartner, Heinz (2004). Regio- and stereoselective reactions of a rhodanine derivative with optically active 2-methyl- and 2-phenyloxirane. Tetrahedron, 60:5407-5412.

Bienz, Stefan; Guggisberg, Armin; Wälchli, Rudolf; Hesse, Manfred (2004). Synthese der Spermidin-Alkaloide (±)-Inandenin-10-ol, Inandenin-10-on und (±)-Oncinotin. Helvetica Chimica Acta, 71(7):1708-1718.

Wälchli, Rudolf; Bienz, Stefan; Hesse, Manfred (2004). Synthese macrocyclischer Lactame aus Ketonen durch Ringerweiterung. Helvetica Chimica Acta, 68(2):484-492.

Bienz, Stefan; Hesse, Manfred (2004). Synthese makrocyclischer Ketone durch Ringerweiterung; ein neuer Weg zu$(\pm)$-Muscon. Helvetica Chimica Acta, 70(8):2146-2151.

Moricz, Attila; Gassmann, Elisabeth; Bienz, Stefan; Hesse, Manfred (2004). Synthesis of $\pm$-pyrenolide B. Helvetica Chimica Acta, 78(3):663-669.

Atanassov, Plamen K; Linden, Anthony; Heimgartner, Heinz (2004). Synthesis of 4-(Phenylamino)quinazoline-2(1H)-selones and Diselenides from Isoselenocyanates: Dimroth Rearrangement of an Intermediate. Helvetica Chimica Acta, 87(7):1873-1887.

Jeremic, Tatjana; Linden, Anthony; Heimgartner, Heinz (2004). Synthesis of Cyclohexapeptides containing Pro and Aib residues. Helvetica Chimica Acta, 87(12):3056-3079.

Smith, Richard J; Bienz, Stefan (2004). Towards Functionalized Silicon-Containingα-Amino Acids: Asymmetric Syntheses of Sila Analogs of Homoserine and Homomethionine. Helvetica Chimica Acta, 87(7):1681-1696.

Tzouros, Manuel; Bigler, Laurent; Bienz, Stefan; Hesse, Manfred; Inada, Akira; Murata, Hiroko; Inatomi, Yuka; Nakanishi, Tsutomu; Darnaedi, Dedy (2004). Two new spermidine alkaloids from Chisocheton weinlandii. Helvetica Chimica Acta, 87(6):1411-1425.


Guintchin, Boris; Bienz, Stefan (2003). Stereoconvergent preparation of chiral vinylsilanes by cuprate substitution of α-acetoxyallylsilanes. Application to the synthesis of ( S )-(+)-bishomomanicone. Tetrahedron, 59(38):7527-7533.

Donath, Marc Y; Störling, Joachim; Maedler, Kathrin; Mandrup-Poulsen, Thomas (2003). Inflammatory mediators and islet ?-cell failure: a link between type 1 and type 2 diabetes. Journal of Molecular Medicine, 81(8):455-470.

Fu, Changchun; Linden, Anthony; Heimgartner, Heinz (2003). 1,3-Oxathiolanes from the reaction of aromatic and enolized thioketones with monosubstituted oxiranes. Helvetica Chimica Acta, 86:2833-2847.

Mekhael, Maged K G; Heimgartner, Heinz (2003). A Novel Synthetic Approach to (±)-Desoxynoreseroline. Helvetica Chimica Acta, 86:2805-2813.

Iliev, Boyan; Linden, Anthony; Heimgartner, Heinz (2003). An unexpected formation of a 14-membered Cyclodepsipeptide. Helvetica Chimica Acta, 86(9):3215-3234.

Stamm, Simon; Linden, Anthony; Heimgartner, Heinz (2003). Chiral Heterospirocyclic 2H-Azirin-3-amines as Synthons for 3-Amino-2,3,4,5-tetrahydrofuran-3-carboxylic Acid and Their Use in Peptide Synthesis. Helvetica Chimica Acta, 86:1371-1396.

Royo, N C; Shimizu, S; Schouten, J W; Stover, J F; McIntosh, T K (2003). Pharmacology of traumatic brain injury. Current Opinion in Pharmacology, 3(1):27-32.

Majchrzak, Agnieszka; Janczak, Aleksandra; Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (2003). Reactions of stable alpha-chlorosulfanyl chlorides with C=S-functionalized compounds. Helvetica Chimica Acta, 86:2272-2283.

Fu, Changchun; Linden, Anthony; Heimgartner, Heinz (2003). Regio- and Stereoselectivity of the SiO2-Catalyzed Reaction of Thiocamphor (= 1,7,7-Trimethylbicyclo[2.2.1]heptane-2-thione) with Optically Active Monosubstituted Oxiranes. Helvetica Chimica Acta, 86:2258-2271.

Atanassov, Plamen K; Linden, Anthony; Heimgartner, Heinz (2003). Selenium-containing heterocycles from Isoselenocyanates: Synthesis of 1H-5-Selena-1,3,6-triazaaceanthrylene derivatives. Helvetica Chimica Acta, 86(9):3235-3243.

Elwan, Nehal M; Awad, Enas M; Hassaneen, Hamdi M; Linden, Anthony; Heimgartner, Heinz (2003). Synthesis of 1,2,4-Triazolo[4,3-a]pyrimidine Derivatives by Cyclocondensation of a 2-Thioxopyrimidin-4(3H)-one with Hydrazonoyl Halides. Helvetica Chimica Acta, 86:739-749.

Luykx, Roeland T N; Linden, Anthony; Heimgartner, Heinz (2003). Synthesis of a Derivative of the Peptaibol-Antibiotic Trichovirin I 1B by means of the 'Azirine/Oxazolone Method'. Helvetica Chimica Acta, 86(12):4093-4111.

Pradeille, Nicolas; Heimgartner, Heinz (2003). Synthesis of the protected 6–16 segment of Zervamicin II-2, an application of the Azirine/Oxazolone method. Journal of Peptide Science, 9(11-12):827-837.


Mlostoń, Grzegorz; Urbaniak, Katarzyna; Heimgartner, Heinz (2002). 1,3-Thiazolidine-dicarboxylates from Thioketones and Thermally Generated Azomethine Ylides. Helvetica Chimica Acta, 85:2056-2064.

Trzoss, Michael; Shao, Jie; Bienz, Stefan (2002). A chiral silyl ether as auxiliary for the asymmetric nucleophilic addition to α- and β-silyloxy carbonyl compounds. Tetrahedron, 58(29):5885-5894.

Breitenmoser, Roland A; Linden, Anthony; Heimgartner, Heinz (2002). Formation of 1,3-Thiazol-5(4H)-imines and 1,3-Oxazol-5(4H)-imines in Aib-Containing Thiopeptides. Helvetica Chimica Acta, 85:990-1018.

Brun, Kathrin A; Linden, Anthony; Heimgartner, Heinz (2002). New Optically Active 2H-Azirin-3-amines as Synthons for Enantiomerically Pure 2,2-Disubstituted Glycines: Synthesis of Synthons for Tyr(2Me) and Dopa(2Me), and Their Incorporation into Dipeptides. Helvetica Chimica Acta, 85:3422-3443.

Awad, Enas M; Elwan, Nehal M; Hassaneen, Hamdi M; Linden, Anthony; Heimgartner, Heinz (2002). New Routes to Fused Isoquinolines. Helvetica Chimica Acta, 85:320-332.

Gendek, Tomasz; Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (2002). Reaction of thiocarbonyl S-methylides with acetylenic dipolarophiles and an unexpected rearrangement of the cycloadducts. Helvetica Chimica Acta, 85:451-463.

Manov, Nikolay; Tzouros, Manuel; Chesnov, Sergiy; Bigler, Laurent; Bienz, Stefan (2002). Solid-Phase Synthesis of Polyamine Spider Toxins and Correlation with the Natural Products by HPLC-MS/MS. Helvetica Chimica Acta, 85(9):2827-2846.

Mlostoń, Grzegorz; Prakash, G K Surya; Olah, George A; Heimgartner, Heinz (2002). Studies on Reactions of Thioketones with Trimethyl(trifluoromethyl)silane Catalyzed by Fluoride Ions. Helvetica Chimica Acta, 85:1644-1658.

Breitenmoser, Roland A; Heimgartner, Heinz (2002). Synthesis and Use of 2H-Azirin-3-amines as Dipeptide Synthons. Helvetica Chimica Acta, 85:885-912.

Atanassov, Plamen K; Zhou, Yuehui; Linden, Anthony; Heimgartner, Heinz (2002). Synthesis of Bis(2,4-diarylimidazol-5-yl) Diselenides from N-Benzylbenzimidoyl Isoselenocyanates. Helvetica Chimica Acta, 85:1102-1117.

Gebert, Andreas; Heimgartner, Heinz (2002). Synthesis of an Enantiomerically Pure 1,3-Thiazole-5(4H)-thione and Its Stereoselective 1,3-Dipolar Cycloaddition with an Azomethine Ylide. Helvetica Chimica Acta, 85:2073-2081.

Mlostoń, Grzegorz; Heimgartner, Heinz (2002). Thiocarbonyl Ylides. In: Padwa, A; Pearson, W H. Synthetic Applications of 1,3-Dipolar Cycloaddition Chemistry Toward Heterocycles and Natural Products. New York: John Wiley & Sons, Inc., 315-360.

Mlostoń, Grzegorz; Urbaniak, Katarzyna; Linden, Anthony; Heimgartner, Heinz (2002). Unexpected Formation of Dimethylthioketene Cycloadducts in the Reaction of 1,3-Diphenylaziridine-2,2-dicarboxylate with Cyclobutanethione Derivatives. Helvetica Chimica Acta, 85:2644-2656.


Hobi, R; Hübscher, U; Neftel, K; Alteri, E; Poncioni, B; Walker, M R; Woods-Cook, K; Schneider, P; Lazdins, J K (2001). Anti-HIV-1 activity in vitro of ceftazidime degradation products. Antiviral Chemistry & Chemotherapy, 12(2):109-118.

Breitenmoser, Roland A; Hirt, Thomas R; Luykx, Roeland T N; Heimgartner, Heinz (2001). A Novel 2H-Azirin-3-amine as a Dipeptide (Aib-Hyp) Synthon. Helvetica Chimica Acta, 84(4):972-979.

Manov, Nikolay; Bienz, Stefan (2001). A new approach in the solid-phase synthesis of polyamine derivatives: construction of polyamine backbones from the center. Tetrahedron, 57(37):7893-7898.

Koch, Kristian N; Hopp, Gudrun; Linden, Anthony; Moehle, Kerstin; Heimgartner, Heinz (2001). Conformational Analysis of the Cyclic Pentadepsipeptide Cyclo(Tro-Aib-Aib-Aib-Aib) in the Solid State and in Solution. Helvetica Chimica Acta, 84(2):502-512.

Brun, Kathrin A; Linden, Anthony; Heimgartner, Heinz (2001). New Optically Active 2H-Azirin-3-amines as Synthons for Enantiomerically Pure 2,2-Disubstituted Glycines. Helvetica Chimica Acta, 84(6):1756-1777.

Fu, Changchun; Linden, Anthony; Heimgartner, Heinz (2001). Regioselectivity of the 1,3-Oxathiolane Formation in the Lewis Acid-Catalyzed Reaction of Thioketones with Asymmetrically Substituted Oxiranes. Helvetica Chimica Acta, 84(11):3319-3334.

Breitenmoser, Roland A; Heimgartner, Heinz (2001). Scope and Limitation of the Acid-Catalyzed Isomerization of Aib-Containing Thiopeptides. Helvetica Chimica Acta, 84(4):786-796.

Awad, Enas M; Elwan, Nehal M; Hassaneen, Hamdi M; Linden, Anthony; Heimgartner, Heinz (2001). Synthesis and Reactivity of 2-(6,7-Diethoxy-3,4-dihydroisoquinolin-1-yl)acetonitrile towards Hydrazonoyl Halides. Helvetica Chimica Acta, 84(5):1172-1180.

Koch, Kristian N; Linden, Anthony; Heimgartner, Heinz (2001). Synthesis of conformationally restricted cyclic pentadepsipeptides via direct amide cyclization. Tetrahedron, 57(12):2311-2326.


Suter, Giovanni; Stoykova, Svetlana A; Linden, Anthony; Heimgartner, Heinz (2000). Heterospirocyclic N-(2H-Azirin-3-yl)-L-prolinates: New Dipeptide Synthons. Helvetica Chimica Acta, 83:2961-2974.

Mlostoń, Grzegorz; Gendek, Tomasz; Heimgartner, Heinz (2000). Reactions of 2-unsubstituted 1H-imidazole 3-oxides with heterocumulenes and dimethyl acetylenedicarboxylate. Tetrahedron, 56:5405-5412.

Zhou, Yuehui; Heimgartner, Heinz (2000). Selenium-containing heterocycles from isoselenocyanates: synthesis of 1,2,3-selenadiazole derivatives. Helvetica Chimica Acta, 83:539-553.

Zhou, Yuehui; Linden, Anthony; Heimgartner, Heinz (2000). Selenium-containing heterocycles from isoselenocyanates: synthesis of 1,3-selenazoles from N-phenylimidoyl isoselenocyanates. Helvetica Chimica Acta, 83:1576-1598.

Blagoev, Milen; Linden, Anthony; Heimgartner, Heinz (2000). Stereochemical course of the reaction between thiocarbonyl compounds and oxiranes: reaction with cis- and trans-2,3-dimethyloxirane. Helvetica Chimica Acta, 83:3163-3178.

Koch, Kristian N; Linden, Anthony; Heimgartner, Heinz (2000). Synthesis of 16-membered cyclic depsipeptides via direct amide cyclization. Helvetica Chimica Acta, 83:233-257.

Koch, Kristian N; Heimgartner, Heinz (2000). Synthesis of conformationally restricted cyclic hexadepsipeptides via direct amide cyclization. Helvetica Chimica Acta, 83:1881-1900.

Mlostoń, Grzegorz; Celeda, Malgorzata; Prakash, G K Surya; Olah, George A; Heimgartner, Heinz (2000). Synthesis of imidazole derivatives using 2-unsubstituted 1H-imidazole 3-oxides. Helvetica Chimica Acta, 83:728-738.


Marx, A; Spichty, M; Amacker, M; Schwitter, U; Hübscher, U; Bickle, T A; Maga, G; Giese, B (1999). Probing interactions between HIV-1 reverse transcriptase and its DNA substrate with backbone-modified nucleotides. Chemistry & Biology, 6(2):111-116.

Lehmann, Jürg; Linden, Anthony; Heimgartner, Heinz (1999). A novel acid-catalyzed isomerization of Aib-containing thiodipeptides. Helvetica Chimica Acta, 82:888-908.

Fässler, Jürg; Enev, Valentin; Bienz, Stefan (1999). A novel stereoselective reaction cascade leading from $\alpha$-silylated allylic alcohols to aldol-type products. Helvetica Chimica Acta, 82(4):561-587.

Muller, J F K; Zehnder, M; Barbosa, F; Spingler, B (1999). Chiral lithiated phosphoric triamides: Structure, reactivity, and salt effects. Helvetica Chimica Acta, 82(9):1486-1501.

Blagoev, Milen; Linden, Anthony; Heimgartner, Heinz (1999). Lewis acid catalyzed reactions of thioketones with 1,2-epoxycyclohexane and 1,2-epoxycyclopentane. Helvetica Chimica Acta, 82:2316-2335.

Pellegrini, N; Refouvelet, B; Crini, G; Blacque, Olivier; Kubicki, M M; Robert, J-F (1999). New dipeptides containing thiazolidine-4-carboxylic acid derivatives: Synthesis and characterization using NMR techniques and X-ray data. Chemical & Pharmaceutical Bulletin, 47(7):950-955.

Blagoev, Milen; Linden, Anthony; Heimgartner, Heinz (1999). Reaction of 1,3-thiazole-5(4H)-thiones with 1,2-epoxycycloalkanes: formation of spirocyclic 1,3-oxathiolanes. Helvetica Chimica Acta, 82:1458-1469.

Mlostoń, Grzegorz; Romański, Jaroslaw; Swia̧tek, Anna; Heimgartner, Heinz (1999). Reactions of thioketones with dichlorocarbene. Helvetica Chimica Acta, 82:946-956.

Todorova, Tonya R; Linden, Anthony; Heimgartner, Heinz (1999). Ring-enlargement and ring-opening reactions of 1,2-thiazetidin-3-one 1,1-dioxides with ammonia and primary amines as nucleophiles. Helvetica Chimica Acta, 82:354-371.

Lehmann, Jürg; Linden, Anthony; Heimgartner, Heinz (1999). Site-selective incorporation of thioamide-linkages into a growing peptide. Tetrahedron, 55:5359-5376.

Fässler, Jürg; Linden, Anthony; Bienz, Stefan (1999). Stereoselective preparation of 2-silylated 1,3-diols and the regioselectivity of their Peterson olefination. Tetrahedron, 55(6):1717-1730.

Lehmann, Jürg; Heimgartner, Heinz (1999). Synthesis of endothiopeptides and their cyclization to 1,3-thiazol-5(4H)-imines. Helvetica Chimica Acta, 82:1899-1915.

Mlostoń, Grzegorz; Gendek, Tomasz; Linden, Anthony; Heimgartner, Heinz (1999). Trapping of a thiocarbonyl ylide with imidazolethiones, pyrimidinethione, and thioamides. Helvetica Chimica Acta, 82:290-296.

Mlostoń, Grzegorz; Romański, Jaroslaw; Linden, Anthony; Heimgartner, Heinz (1999). Unexpected products from the reaction of 2,2,4,4-tetramethylcyclobutane-1,3-dione with the Makosza reagent. Helvetica Chimica Acta, 82:1302-1310.


Hoepping, A; Reisgys, M; Brust, P; Seifert, S; Spies, H; Alberto, R; Johannsen, B (1998). TROTEC-1: a new high-affinity ligand for labeling of the dopamine transporter. Journal of Medicinal Chemistry, 41(23):4429-4432.

von Janta-Lipinski, M; Costisella, B; Ochs, H; Hübscher, U; Hafkemeyer, P; Matthes, E (1998). Newly synthesized L-enantiomers of 3'-fluoro-modified beta-2'-deoxyribonucleoside 5'-triphosphates inhibit hepatitis B DNA polymerases but not the five cellular DNA polymerases alpha, beta, gamma, delta, and epsilon nor HIV-1 reverse transcriptase. Journal of Medicinal Chemistry, 41(12):2040-2046.

Perrin, Sandrine; Monnier, Karin; Laude, Bernard; Kubicki, Marek M; Blacque, Olivier (1998). Reaction of an open-chain analogue of Reissert compound hydrofluoroborate salt with ethyl acrylate. A reinvestigation. Tetrahedron Letters, 39(13):1753-1754.

Kägi, Martin; Linden, Anthony; Mlostoń, Grzegorz; Heimgartner, Heinz (1998). 1,3-Oxathiole and Thiirane Derivatives from the Reactions of Azibenzil and alpha-Diazo Amides with Thiocarbonyl Compounds. Helvetica Chimica Acta, 81(2):285-302.

Moya Argilagos, Dally; Kunz, Roland W; Linden, Anthony; Heimgartner, Heinz (1998). Desulfurization of 4-Nitro-N,2-diphenyl-3-(phenylamino)isothiazol-5(2H)-imine: Formation of a 3-Imino-2-nitroprop-2-enamidine. Helvetica Chimica Acta, 81(12):2388-2406.

Mlostoń, Grzegorz; Gendek, Tomasz; Heimgartner, Heinz (1998). First examples of reactions of azole n-oxides with thioketones: a novel type of sulfur-transfer reaction. Helvetica Chimica Acta, 81(9):1585-1595.

Peghini, P A; Zahner, R; Kuster, H; Schott, H; Schwendener, R (1998). In vitro anti-human immunodeficiency virus and anti-hepatitis B virus activities and pharmacokinetic properties of heterodinucleoside phosphates containing AZT or ddC. Antiviral Chemistry & Chemotherapy, 9(2):117-126.

Garcia Trimino, Maria I; Macias Cabrera, Arturo; Velez Castro, Herman; Rosado Perez, Aristide; Moya Argilagos, Dally; Linden, Anthony; Heimgartner, Heinz (1998). Reaction of N,N'-Dimethyl-2-nitroethene-1,1-diamine with alpha,beta-Unsaturated Acyl Isothiocyanates: Preparation of 1,3-Thiazin-4-one and 4-Nitro-1,2-thiazol-5(2H)-imine Derivatives. Helvetica Chimica Acta, 81(3-4):718-728.

Lehmann, Jürg; Linden, Anthony; Heimgartner, Heinz (1998). Synthesis of the Endothiopeptide BOC-Trp-Ile-Ala-Aib-lle-Val[CSNH]Aib-Leu-Aib-Pro-OMe by a Variation of the 'Azirine/Oxazolone Method'. Tetrahedron, 54(30):8721-8736.

van Borssum Waalkes, M; Goris, H; Dontje, B H; Schwendener, R; Scherphof, G; Nijhof, W (1998). Toxicity of liposomal 3'-5'-O-dipalmitoyl-5-fluoro-2'-deoxyuridine in mice. Anti-Cancer Drug Design, 13(4):291-305.

Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (1998). [2+3] Cycloadditions of Azomethine Ylides with 1,3-Thiazole-5(4H)-thiones. Helvetica Chimica Acta, 81(3-4):558-569.


Jentgens, Christian; Bienz, Stefan; Hesse, Manfred (1997). Selective monoderivatization of propane-1,3-diamine with acid chlorides: ‘Hexahydropyrimidine method’ vs. statistic methods. Helvetica Chimica Acta, 80(4):1133-1143.

Mlostoń, Grzegorz; Romański, Jaroslaw; Linden, Anthony; Heimgartner, Heinz (1997). "Three-Component reaction" with aromatic thioketones, phenyl azide, and dimethyl fumarate. Helvetica Chimica Acta, 80:1992-2001.

Meier, Karl-Richard; Linden, Anthony; Mlostoń, Grzegorz; Heimgartner, Heinz (1997). 1,3-dipolare Cycloadditionen eines Carbonyl-ylids mit 1,3-Thiazol-5(4H)-thionen und Thioketonen. Helvetica Chimica Acta, 80:1190-1204.

Moya Argilagos, Dally; Garcia Trimino, Maria I; Macias Cabrera, Arturo; Linden, Anthony; Heimgartner, Heinz (1997). An unexpected isomerization of N-Aryl-3-amino-4-nitroisothiazol-5(2H)-imines to 2-(Benzothiazol-2-y1)-2-nitroethene-1,1-diamines. Helvetica Chimica Acta, 80:273-292.

Strässler, Christof; Heimgartner, Heinz (1997). An unexpected transformation of benzyl carbamates into alpha-azidobenzeneacetamides. Helvetica Chimica Acta, 80:2058-2065.

Strässler, Christof; Linden, Anthony; Heimgartner, Heinz (1997). Novel heterospirocyclic 3-amino-2H-azirines as synthons for heterocyclic alpha-amino acids. Helvetica Chimica Acta, 80:1528-1554.

Mlostoń, Grzegorz; Romański, Jaroslaw; Linden, Anthony; Heimgartner, Heinz (1997). Ringöffnungen von sterisch gehinderten spirocyclischen 2,5-Dihydro- 1,3,4-thiadiazolen mit cycloaliphatischen, sekundären Aminen. Helvetica Chimica Acta, 80:230-240.

Jentgens, Christian; Hofmann, Richard; Guggisberg, Armin; Bienz, Stefan; Hesse, Manfred (1997). Selective synthesis of polyamine derivatives: Efficient derivatization of the secondary amino group ofN-monosubstituted 1,3-diamines. Helvetica Chimica Acta, 80(3):966-978.

Villalgordo, Jose M; Heimgartner, Heinz (1997). Synthesis of cyclic depsipeptides and peptides via direct amide cyclization. Helvetica Chimica Acta, 80:748-766.

Smith, Richard J; Bratovanov, Svetoslav; Bienz, Stefan (1997). Synthesis of silicon-containing α-amino acids and hydantoins. Tetrahedron, 53(40):13695-13702.


Meyers, Albert I; Bienz, Stefan; Kwon, Hyok-Boong; Wallace, Richard H (1996). The asymmetric synthesis of fused cyclopentenone ring systems: a formal asymmetric total synthesis of (−)-isocomene. Helvetica Chimica Acta, 79(4):1026-1046.

Enev, Valentin; Stojanova, Diana; Bienz, Stefan (1996). Chiral Acylsilanes in Organic Synthesis. Part 3. Silicon-directed stereoselective preparation and Ireland ester-enolate rearrangement of O-acyl-substituted α-silylated allyl alcohols. Helvetica Chimica Acta, 79(2):391-404.

Kägi, Martin; Linden, Anthony; Mlostoń, Grzegorz; Heimgartner, Heinz (1996). 1,5-Dipolare Elektrocyclisierung von Acyl-substituierten ‘Thiocarbonyl-yliden’ zu 1,3-Oxathiolen. Helvetica Chimica Acta, 79(3):855-874.

Villalgordo, Jose M; Linden, Anthony; Heimgartner, Heinz (1996). A novel amination reaction with Diphenyl Phosphorazidate: Synthesis of alpha-Amino-Acid Derivatives. Helvetica Chimica Acta, 79(1):213-219.

Orahovats, Alexander S; Bratovanov, Svetoslav B; Linden, Anthony; Heimgartner, Heinz (1996). A ring enlargement from seven- to ten-membered-ring sulfonamide derivatives. Helvetica Chimica Acta, 79(4):1121-1128.

Mlostoń, Grzegorz; Heimgartner, Heinz (1996). Carbenoid reactions of Dimethyl Diazomalonate with aromatic Thioketones and 1,3-Thiazole-5(4H)-thiones. Helvetica Chimica Acta, 79(7):1785-1792.

Luykx, Roeland; Bucher, Christoph B; Linden, Anthony; Heimgartner, Heinz (1996). Ein neues 3-Amino-2H-azirin als Aib-Pro-Baustein: Synthese des C-terminalen Nonapeptids von Trichovirin I 1B. Helvetica Chimica Acta, 79(2):527-540.

Shi, Junxing; Heimgartner, Heinz (1996). New addition reactions of organometal compounds with 4,4-Dimethyl-1,3-thiazole-5(4H)-thione. Helvetica Chimica Acta, 79(2):371-384.

Bucher, Christoph B; Heimgartner, Heinz (1996). Optisch aktive 3-Amino-2H-azirine als Bausteine für enantiomerenreine alpha,alpha-disubstituierte alpha-Aminosäuren: Synthese von Isovalin-Synthonen und Einbau in ein Trichotoxin-A-50-Segment. Helvetica Chimica Acta, 79(7):1903-1915.

Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (1996). Regioselektive 1,3-Dipolare Cycloadditionen eines ‘Thiocarbonyl-methanids’ ((Alkylidensulfonio)methanids) mit aromatischen Sulfinen. Helvetica Chimica Acta, 79(1):31-40.

Muller, J F K; Batra, R; Spingler, B; Zehnder, M (1996). Synthesis and X-ray structure of bis{S-(1-lithio-3,3-diphenylprop-2-enyl)-N-methyl-S-phenylsulfoximine-t etrahydrofuran(1/2)} complemented by model ab initio calculations of alpha-lithiosulfoximines. Helvetica Chimica Acta, 79(3):820-826.

Schott, H; Schwendener, R (1996). Synthesis and structure-activity studies in vivo of liposomal phospholipid-N4-palmitoyl- and N4-hexadecyl-1-beta-D-arabinofuranosylcytosine conjugates. Anti-Cancer Drug Design, 11(6):451-62.

Mihova, Tonya R; Linden, Anthony; Heimgartner, Heinz (1996). Synthesis of 1,2,5-Thiadiazepine Derivatives by Ring Enlargement of 1,2-Thiazetidin-3-one 1,1-Dioxides with 3-Amino-2H-azirines. Helvetica Chimica Acta, 79(8):2067-2074.

Mlostoń, Grzegorz; Romański, Jaroslaw; Linden, Anthony; Heimgartner, Heinz (1996). Three-component reactions with Sterically Crowded 2,2,4,4-Tetramethyl-3-thioxocyclobutanone, Phenyl Azide, and Electron-Deficient C,C-Dipolarophiles. Helvetica Chimica Acta, 79(5):1305-1314.

Aguzzi, A; Brandner, S; Marino, S; Steinbach, J P (1996). Transgenic and knockout mice in the study of neurodegenerative diseases. Journal of Molecular Medicine, 74(3):111-126.


Hugener, Martin; Heimgartner, Heinz (1995). 4-Amino-1,5-dihydro-2H-pyrrol-2-one aus Bortrifluorid-katalysierten Umsetzungen von 3-Amino-2H-azirinen mit Carbonsäure-Derivaten. Helvetica Chimica Acta, 78:1490-1498.

Villalgordo, Jose M; Enderli, Adelheid; Linden, Anthony; Heimgartner, Heinz (1995). Diazo-transfer reaction with diphenyl phosphorazidate. Helvetica Chimica Acta, 78:1983-1998.

Hugener, Martin; Heimgartner, Heinz (1995). Eine überraschende Ringerweiterung von 3-(Dimethylamino)-2,2-dimethyl-2H-azirin zu 4,5-Dihydropyridin-2(3H)-on-Derivaten. Helvetica Chimica Acta, 78:1863-1878.

Mlostoń, Grzegorz; Romański, Jaroslaw; Linden, Anthony; Heimgartner, Heinz (1995). Erstes Beispiel einer H-Verschiebung in ‘Thiocarbonyl-aminiden’(N-(Alkylidensulfonio)aminiden). Helvetica Chimica Acta, 78:1067-1078.

Bucher, Christoph B; Linden, Anthony; Heimgartner, Heinz (1995). Optisch aktive 3-Amino-2H-azirine als Bausteine für enantiomerenreine alpha,alpha-disubstituierte alpha-Aminosäuren: Synthese des alpha-Methylphenylalanin-Synthons and Einbau in Modell-Peptide. Helvetica Chimica Acta, 78:935-946.

Huber, Priska; Enev, Valentin; Linden, Anthony; Bienz, Stefan (1995). The reaction of acylsilane-enolates with benzaldehyde: Reaction cascade leading to α-Benzoyloxy-γ-hydroxysilanes. Tetrahedron, 51(13):3749-3754.


Magirius, Florian; Linden, Anthony; Heimgartner, Heinz (1994). 4,4-Disubstituierte Imidazol-Derivate aus der Umsetzung von 3-Amino-2H-azirinen mit Salicylamid. Helvetica Chimica Acta, 77(2):453-462.

Petit, Mireille; Linden, Anthony; Mlostoń, Grzegorz; Heimgartner, Heinz (1994). Reaktion von Phenyldiazomethan mit 1,3-Thiazol-5(4H)-thionen: Basenkatalysierte Ring-Öffnung des Primäradduktes. Helvetica Chimica Acta, 77(4):1076-1086.

Shi, Junxing; Tromm, Peter; Heimgartner, Heinz (1994). Synthesis and addition reactions of 1,3-Thiazole-5(4H)-thione Oxides. Helvetica Chimica Acta, 77:2133-2141.

Shi, Yunxing; Linden, Anthony; Heimgartner, Heinz (1994). Synthesis and reactions of 2-(Alkylthio)-4,4-dimethyI-1,3-thiazole-5(4H)-thiones. Helvetica Chimica Acta, 77(7):1903-1920.

Bienz, Stefan; Enev, Valentin; Huber, Priska (1994). Synthesis of 4(benzyloxymethyl)(tert.-butyl)methylsilyloxy-1,2,3-pentatriene via Brook rearrangement. Tetrahedron Letters, 35(8):1161-1162.

Hadj-Abo, Ferrid; Bienz, Stefan; Hesse, Manfred (1994). Synthesis of [10]heterophanes using a ring enlargement reaction. Tetrahedron, 50(29):8665-8672.

Meier, Hans Rudolf; Heimgartner, Heinz (1994). Tetrazoles. In: Schaumann, Ernst. Methoden der Organischen Chemie (Houben-Weyl). Stuttgart, Germany: Georg Thieme Verlag, 664-795.

Mlostoń, Grzegorz; Petit, Mireille; Linden, Anthony; Heimgartner, Heinz (1994). Umsetzung von Di(tert-buty1)- und Diphenyldiazomethan mit 1,3-Thiazol-5(4H)-thionen: Isolierung und Kristallstruktur des primären Cycloadduktes. Helvetica Chimica Acta, 77(2):435-444.

Kägi, Martin; Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (1994). Umsetzung von Diazoessigsäure-ethylester mit 1,3-Thiazol-5(4H)-thionen. Helvetica Chimica Acta, 77(5):1299-1312.


Chapeaurouge, Alexander; Bienz, Stefan (1993). Chiral acylsilanes in organic synthesis. Part 2. The role of the solvent, the organometallic reagent, and the nature of the substrate for the diastereoselectivity of 1,2-additions to racemic alkoxymethyl-substituted acylsilanes. Helvetica Chimica Acta, 76(5):1876-1889.

Matile, Stefan; Janowitz, Agnes; Ghirlanda, Sandro; Lorenzi-Riatsch, Annalaura; Horni, Albert; Moricz, Attila; Bienz, Stefan; Bild, Norbert; Woggon, Wolf-Dietrich; Hesse, Manfred (1993). Nachbargruppeneffekte in der Gas-Phase: Intramolekulare Deacetalisierung von Hydroxyacetalen unter den Bedingungen der chemischen Ionisation. Helvetica Chimica Acta, 76(3):1305-1310.

Garcia Trimino, Maria I; Linden, Anthony; Heimgartner, Heinz; Macias Cabrera, Arturo (1993). 3-(Acylamino)-3-amino-2-nitroacrylonitriles from N-Acyl-S-methyl-3,3-diamino-2-nitroacrylthioimidates. Helvetica Chimica Acta, 76:2817-2829.

Mütsch, Margot; Erdelmeier, C A J; Sticher, O; Reuter, H D (1993). A Novel Amino Acid Glycoside and Three Amino Acids from Allium sativum. Journal of natural products, 56(6):864-869.

Villalgordo, Jose M; Heimgartner, Heinz (1993). A Novel Synthesis of 2,2-Disubstituted 3-Amino-2H-azirines Based on the Reaction between Amide Enolates and Diphenyl Phosphorochloridate. Helvetica Chimica Acta, 76:2830-2837.

Heimgartner, Heinz; Hansen, Hans-Jürgen (1993). Organische Photochemie im Spiegel von Helvetica Chimica Acta. Helvetica Chimica Acta, 76:1027-1114.

Schläpfer-Dähler, Marlise; Heimgartner, Heinz (1993). Ring-Transformationen bei der Umsetzung von 3-(Dimethylamino)-2,2-dimethyl-2H-azirin mit 1-substituierten Imidazolidin-2,4,5-trionen. Helvetica Chimica Acta, 76:2321-2328.

Kägi, Martin; Linden, Anthony; Heimgartner, Heinz; Mlostoń, Grzegorz (1993). Umsetzung von 1,3-Thiazol-5(4H)-thionen mit Diazomethan. Helvetica Chimica Acta, 76:1715-1728.

Magirius, Florian; Linden, Anthony; Heimgartner, Heinz (1993). Umsetzung von 3-Amino-2H-azirinen mit Salicylohydrazid. Helvetica Chimica Acta, 76:1980-2003.

Villalgordo, Jose M; Heimgartner, Heinz (1993). Synthesis of a Novel Heterospirocyclic 3-(N-Methyl-N-phenylamino)-2H-azirine and its Use as an Amino Acid Equivalent in the Preparation of a Model Tripeptide. Tetrahedron, 49:7215-7222.


Obrecht, Daniel; Spiegler, Clive; Schönholzer, Peter; Müller, Klaus; Heimgartner, Heinz; Stierli, Friedrich (1992). A New General Approach to Enantiomerically Pure Cyclic and Open-Chain (R) - and (S)-alpha,alpha-Disubstituted alpha-Amino Acids. Helvetica Chimica Acta, 75:1666-1696.

Orahovats, Alexander S; Linden, Anthony; Heimgartner, Heinz (1992). A Ring-Enlargement Reaction Yielding 1,2,5-Benzothiadiazonin-6-one 1,1-Dioxides. Helvetica Chimica Acta, 75:2515-2519.

Trifonov, Latchezar S; Orahovats, Alexander S; Linden, Anthony; Heimgartner, Heinz (1992). Carbonyliron Complexation and Carbonyl Insertion of Allenic Ketones. Helvetica Chimica Acta, 75:1872-1879.

Villalgordo, Jose M; Heimgartner, Heinz (1992). Reaction of Diphenyl Phosphorochloridate with Amide Enolates: A New and Convenient Synthesis of 2-Monosubstituted 3-(N-Methyl-N-phenylamino)-2H-azirines. Helvetica Chimica Acta, 75:1866-1871.

Villalgordo, Jose M; Linden, Anthony; Heimgartner, Heinz (1992). Reactions of 2-Monosubstituted 3-Amino-2H-azirines with NH-Acidic Heterocycles. Helvetica Chimica Acta, 75:2270-2282.

Mlostoń, Grzegorz; Heimgartner, Heinz (1992). Reaktion von 2-Diazopropan mit 1,3-Thiazol-5(4H)-thionen. Helvetica Chimica Acta, 75:1825-1833.

Schläpfer-Dähler, Marlise; Mukherjee-Müller, Gabriele; Heimgartner, Heinz (1992). Ring-Transformation von Imidazolidin-2,4-dionen (= Hydantoinen) zu 4H-Imidazolen bei der Umsetzung mit 3-(Dimethylamino)-2,2-dimethyl-2H-azirin. Helvetica Chimica Acta, 75:1251-1261.

Heimgartner, Heinz; Hansen, Hans-Jürgen (1992). Struktur und Mechanismus in der organischen Chemie im Spiegel von Helvetica Chimica Acta. Helvetica Chimica Acta, 75(2):359-437.


Oremus, Vladimir; Linden, Anthony; Heimgartner, Heinz (1991). 1,3-Oxathiolan-Synthese: Spirocyclische 1,3-Oxathiolane aus der Lewis-Säure-katalysierten Umsetzung von cyclischen Trithiocarbonaten und Oxiranen. Helvetica Chimica Acta, 74(7):1500-1510.

Bienz, Stefan; Chapeaurouge, Alexander (1991). Chiral Acylsilanes in Organic Synthesis. Diastereoselective 1,2-Additions to Racemic Alkoxymethyl-Substituted Acylsilanes. Helvetica Chimica Acta, 74(7):1477-1488.

Mihova, Tonya R; Trifonov, Latchezar S; Dimitrov, Valentin S; Orahovats, Alexander S; Linden, Anthony; Heimgartner, Heinz (1991). New Polycyclic Compounds from Photochemical Rearrangements of Some Substituted 2-Azatricyclo[]undeca-4,8,10-trien-3-ones. Helvetica Chimica Acta, 74(5):1011-1026.

Mlostoń, Grzegorz; Linden, Anthony; Heimgartner, Heinz (1991). Regioselektive 1,3-dipolare Cycloadditionen von Thiocarbonyl-yliden mit 1,3-Thiazol-5(4H)-thionen. Helvetica Chimica Acta, 74(7):1386-1398.

Rahm, Annette; Linden, Anthony; Vincent, Beverly R; Heimgartner, Heinz; Mühlstädt, Manfred; Schulze, Bärbel (1991). Ringerweiterung von 1,2-Thiazol-3(2H)-on-1,1-dioxiden und 3-Amino-2H-azirinen zu 4H-1,2,5-Thiadiazocin-6-on-1,1-dioxiden. Helvetica Chimica Acta, 74(5):1002-1010.

Schulze, Bärbel; Kirsten, Gisela; Kirrbach, Sabine; Rahm, Annette; Heimgartner, Heinz (1991). Zur Oxidation von 1,2-Thiazolen: Ein einfacher Zugang zu 1,2-Thiazol-3(2H)-on-1,1-dioxiden. Helvetica Chimica Acta, 74(5):1059-1070.


Trifonov, Latchezar S; Orahovats, Alexander S; Heimgartner, Heinz (1990). Carbonyliron Complexes of Allenic Acids, Esters, Amides, and Imides. Helvetica Chimica Acta, 73(6):1734-1741.

Ametamey, Simon M; Vincent, Beverly R; Heimgartner, Heinz (1990). Dipolare (1:1)-Addukte aus der Reaktion von 3-Amino-2H-azirinen mit 1,3,4-Oxadiazol- und 1,3,4-Thiadiazol-2(3H)-onen. Helvetica Chimica Acta, 73(2):492-507.

Tromm, Peter-Claus; Heimgartner, Heinz (1990). Eine neue 1,3-Oxathiolan-Synthese: Spirocyclische 1,3-0xathiolane aus der Lewis-Säure katalysierten Umsetzung von 1,3-Thiazol-5(4H)-thionen mit Oxiranen. Helvetica Chimica Acta, 73(8):2287-2294.

Villalgordo, Jose M; Vincent, Beverly R; Heimgartner, Heinz (1990). Reaction of 3-Amino-2H-azirines with 2-Amino-4,6-dinitrophenol (Picramic Acid): Synthesis of Quinazoline- and 1,3-Benzoxazole Derivatives. Helvetica Chimica Acta, 73(4):959-974.

Ametamey, Simon M; Heimgartner, Heinz (1990). Reaktionen von 3-(Dimethylamino)-2H-azirinen mit 1,3-Benzoxazol-2(3H)-thion. Helvetica Chimica Acta, 73(3):599-607.

Ametamey, Simon M; Heimgartner, Heinz (1990). Ringerweiterungen und Ringverengungen bei der Umsetzung von 1,3- Oxazolidin-2,4-dionen und 1,3-Thiazolidin-2,4-dion mit 3-Amino-2H-azirinen. Helvetica Chimica Acta, 73(5):1314-1328.

Obrecht, Daniel; Heimgartner, Heinz (1990). Synthese cyclischer Depsipeptide durch direkte Amid-Cyclisierung: 12gliedrige Depsipeptide mit alternierender Sequenz von α-Hydroxy- und α-Aminosäuren. Helvetica Chimica Acta, 73(1):221-228.

Wipf, Peter; Heimgartner, Heinz (1990). Synthesis of Peptides Containing alpha,alpha-Disubstituted alpha-Amino Acids by the Azirine/Oxazolone Method: The (12-20)-Nonapeptide of the Ionophore Alamethicin. Helvetica Chimica Acta, 73(1):13-24.

Ametamey, Simon M; Heimgartner, Heinz (1990). Umsetzung von 3-(Dimethylamino)-2H-azirinen mit 1,3-Oxazolidin-2-thion zu 3-(2-Hydroxyethyl)-2-thiohydantoinen. Helvetica Chimica Acta, 73(3):594-598.

Schläpfer-Dähler, Marlise; Heimgartner, Heinz (1990). Umsetzungen von 3-(Dimethylamino)-2,2-dimethyl-2H-azirim mit Barbitursäure-Derivaten. Helvetica Chimica Acta, 73(8):2275-2286.


Sahebi, Mostafa; Wipf, Peter; Heimgartner, Heinz (1989). 3-amino-2h-azirines in the synthesis of peptides: tetrapeptides with alpha,alpha-disubstituted alpha-amino acids. Tetrahedron, 45(10):2999-3010.

Jenny, Christjohannes; Heimgartner, Heinz (1989). Bildung von 5,6-Dihydro-1,3(4H)-thiazin-4-carbonsäure-estern aus 4-Allyl-1,3-thiazol-5(4H)-onen. Helvetica Chimica Acta, 72:1639-1646.

Hugener, Martin; Heimgartner, Heinz (1989). Eine neue Aminoazirin-Reaktion. Bildung von 3,6-Dihydropyrazin-2(1H)-onen. Helvetica Chimica Acta, 72:172-179.

Jenny, Christjohannes; Wipf, Peter; Heimgartner, Heinz (1989). Radikalische Cyclisierungen von Alkenyl-substituierten 4,5-Dihydro-1,3-thiazol-5-thiolen. Helvetica Chimica Acta, 72:838-846.

Bozhkova, Nina; Heimgartner, Heinz (1989). Synthesis of 4-Alkoxy-1,3-oxazol-5(2H)-ones, Precursors of 1-Alkoxy-Substituted Nitrile Ylides. Helvetica Chimica Acta, 72:825-837.


Wipf, Peter; Prewo, Roland; Bieri, Jost H; Germain, Gabriel; Heimgartner, Heinz (1988). (Benzylthio)- und (Arylthio)-substituierte Nitril-ylide: thermische Erzeugung und Reaktionen. Helvetica Chimica Acta, 71(5):1177-1190.

Ametamey, Simon M; Hollenstein, Roger; Heimgartner, Heinz (1988). 15N-Markiertes 3-(Dimethylamino)-2,2-dimethyl-2H-azirin zur mechanistischen Untersuchung von Reaktionen rnit NH-aciden Heterocyclen. Helvetica Chimica Acta, 71(3):521-530.

Wipf, Peter; Heimgartner, Heinz (1988). Anwendung der Azirin/Oxazolon-Methode in der Peptid-Chemie: Synthese von Modell-Tripeptiden. Helvetica Chimica Acta, 71(1):140-154.

Tromm, Peter; Heimgartner, Heinz (1988). Hetero-Diels-Alder-Reaktion mit 1,3-Thiazol-5(4H)-thionen. Helvetica Chimica Acta, 71(8):2071-2084.

Wipf, Peter; Heimgartner, Heinz (1988). Konformationsanalysen von Modell-Tripeptiden: Der Einfluss von alpha,alpha-disubstituierten alpha-Aminosäuren auf die Sekundärstruktur. Teil I: NMR- und CD-Untersuchungen. Helvetica Chimica Acta, 71(1):258-267.

Wipf, Peter; Kunz, Roland W; Prewo, Roland; Heimgartner, Heinz (1988). Konformationsanalysen von Modell-Tripeptiden: Der Einfluss von alpha,alpha-disubstituierten alpha-Aminosäuren auf die Sekundärstruktur. Teil II. Röntgenstrukturanalyse und Konformationsenergie-Berechnungen. Helvetica Chimica Acta, 71(1):268-273.

Pekcan, Sare; Heimgartner, Heinz (1988). N-(1,3-Thiazol-5(4H)-yliden)amine aus 1,3-dipolaren Cycloadditionen von Aziden mit 1,3-Thiazo1-5(4H)-thionen. Helvetica Chimica Acta, 71(7):1673-1680.

Trifonov, Latchezar S; Orahovats, Alexander S; Prewo, Roland; Heimgartner, Heinz (1988). Synthesis and Structure of Carbonyliron Complexes of Allenecarboxylates and Allenic Lactones. Helvetica Chimica Acta, 71(3):551-561.

Obrecht, Jean-Pierre; Schönholzer, Peter; Jenny, Christian Johannes; Prewo, Roland; Heimgartner, Heinz (1988). The Reaction of 3-(Dimethylamino)-2H-azirines with 2,3-Pyridinedicarboximide. Helvetica Chimica Acta, 71(5):1319-1327.


Obrecht, Daniel; Heimgartner, Heinz (1987). 3-(Dimethylamino)-2,2-dimethyl-2H-azirin als Aib-Äquivalent: Synthese von Aib-Oligopeptiden. Helvetica Chimica Acta, 70:102-115.

Obrecht, Daniel; Heimgartner, Heinz (1987). 3-(Dimethylamino)-2,2-dimethyl-2H-azirin als alpha-Aminoisobuttersäure (Aib)-Aquivalent: Cyclische Depsipeptide durch direkte Amid-Cyclisierung. Helvetica Chimica Acta, 70:329-338.

Wipf, Peter; Heimgartner, Heinz (1987). Bildung tricyclischer Thietan-Derivate durch intramolekulare (2+2)-Cycloaddition. Helvetica Chimica Acta, 70:992-994.

Trifonov, Latchezar S; Orahovats, Alexander S; Heimgartner, Heinz (1987). Octacarbonyldicobalt-Induced (1,3) H Shifts in 1-Methylallenecarboxylates and Allenic Lactones. Helvetica Chimica Acta, 70:1070-1075.

Wipf, Peter; Heimgartner, Heinz (1987). Selektive Amidspaltung bei Peptiden mit alpha,alpha-disubstituierten alpha-Aminosäuren. Helvetica Chimica Acta, 70:354-368.

Bienz, Stefan; Hesse, Mauhad (1987). Synthese makrocyclischer, $\alpha, \beta$-ungesättigter y-Oxolactone durch Ringerweiterungsreaktionen; ein neuer Weg zum makrocyclischen Lacton-Antibiotikum A 26771 B. Helvetica Chimica Acta, 70(5):1333-1340.

Wipf, Peter; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz; Nastopoulos, Vassilios; Germain, Gabriel (1987). Synthese von 4-Benzylthio- und 4-(Arylthio)-1,3-oxazol-5(2H)-onen. Helvetica Chimica Acta, 70:1380-1388.


Jenny, Christjohannes; Heimgartner, Heinz (1986). 1,4-Dithiafulvene aus der Umsetzung von 4,4-disubstituierten 1,3-Thiazol-5(4H)-thionen mit Acetylenderivaten. Helvetica Chimica Acta, 69(2):419-429.

Hostettler, Bernhard; Obrecht, Jean-Pierre; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz (1986). 5,6,7,8-Tetrahydro-4H-1,2,5-oxadiazocin-6-one durch Ringerweiterung nach Addition eines 3-lsoxazolidinons mit 3-Amino-2H-azirinen. Helvetica Chimica Acta, 69(2):298-304.

Jenny, Christjohannes; Heimgartner, Heinz (1986). Additionsreaktion von 1,3-Thiazol-5(4H)-thionen und Inaminen; Bildung von Thioamiden und Thioketonen. Helvetica Chimica Acta, 69(1):174-183.

Jenny, Christjohannes; Wipf, Peter; Heimgartner, Heinz (1986). Carbophile Additionen von Organocupraten mit 1,3-Thiazo1-5(4H)-thionen. Helvetica Chimica Acta, 69(8):1837-1843.

Wipf, Peter; Heimgartner, Heinz (1986). Kupplung von Peptiden mit C-terminalen alpha,alpha-disubstituierten alpha-Aminosäuren via Oxazol-5(4H)-one. Helvetica Chimica Acta, 69(5):1153-1162.

Ametamey, Simon M; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz; Obrecht, Jean-Pierre (1986). Reaktion von 3-(Dimethylamino)-2H-azirinen mit 1,3-Thiazolidin-2-thion. Helvetica Chimica Acta, 69(8):2013-2025.

Jenny, Christjohannes; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz (1986). Synthese von (Methylthio)penam-Derivaten durch Keten-Addition an 4,5-Dihydro-5-(methylthio)-1,3-thiazole. Helvetica Chimica Acta, 69(6):1424-1434.

Jenny, Christjohannes; Heimgartner, Heinz (1986). Synthese von 4,4-disubstituierten 1,3-ThiazoI-5(4H)-thionen. Helvetica Chimica Acta, 69(2):374-388.

Jenny, Christjohannes; Heimgartner, Heinz (1986). Umsetzungen von 1,3-Thiazol-5(4H)-thionen mit Grignard- und Organolithium-Verbindungen: Carbophile und Thiophile Additionen. Helvetica Chimica Acta, 69(4):773-785.

Meier, Hansruedi; Heimgartner, Heinz (1986). lntramolekulare 1,3-dipolare Cycloadditionen mit alkenyl-substituierten 3,4-Diarylsydnonen. Helvetica Chimica Acta, 69(4):927-940.


Meier, Hansruedi; Heimgartner, Heinz (1985). Intramolekulare 1,3-dipolare Cycloadditionen von Diarylnitriliminen aus 2,5-Diaryltetrazolen. Helvetica Chimica Acta, 68(5):1283-1300.

Obrecht, Daniel; Scholl, Bernhard; Heimgartner, Heinz (1985). Synthese von 3,3-Dimethylperhydro-1,4-diazepin-2,5,7-trionen aus 3-Dimethylamino-2,2-dimethyl-2H-azirin und Malonsäuremonoamiden. Helvetica Chimica Acta, 68(2):465-474.

Lukac, Josef; Heimgartner, Heinz (1985). Umlagerungsreaktionen von (2’-Propinyl)cyclohexadienolen und -semibenzolen. Helvetica Chimica Acta, 68(2):355-370.


Büchel, Thomas; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz (1984). 1,3-Dipolare Cycloadditionen von Nitrilium-Betainen mit 4,4-Dimethyl-2-phenyl-2-thiazolin-5-thion. Helvetica Chimica Acta, 67:534-549.

Obrecht, Daniel; Heimgartner, Heinz (1984). Eine neue Lactonsynthese via 2-Oxazolin-5-one als Zwischenprodukte. Tetrahedron Letters, 25(16):1717-1720.

Obrecht, Daniel; Heimgartner, Heinz (1984). Synthese eines cyclischen Depsipeptides mittels Amidcyclisierung. Helvetica Chimica Acta, 67:526-533.

Stierli, Friedrich; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz (1984). Synthese und Struktur von Zink-Komplexen von 2-Amino-1-azetinen. Helvetica Chimica Acta, 67:927-933.

Wipf, Peter; Heimgartner, Heinz (1984). Synthese von 4-Arylthio-3-oxazolin-5-onen. Tetrahedron Letters, 25(45):5127-5128.


Obrecht, Daniel; Heimgartner, Heinz (1983). 3-dimethylamino-2,2-dimethyl-2h-azirin als aib-aequivalent bei heterocyclen-synthesen; synthese von 6-, 9-, 12- und 15-gliedrigen ringen. Tetrahedron Letters, 24(18):1921-1924.

Stierli, Friedrich; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz (1983). Additionsreaktionen von 2-Amino-1-azetinen mit Cyclopropenonen; Bildung von Azepinderivaten durch Ringerweiterung. Helvetica Chimica Acta, 66:1366-1375.

Dähler, Marlise; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz (1983). Heterocyclole als Zwischenprodukte einer neuen, überraschenden Umlagerung bei der Reaktion von 3-(Dimethylamino)-2,2-dimethyl-2H-azirin mit monosubstituierten Parabansäuren. Helvetica Chimica Acta, 66:1456-1465.

Dietliker, Kurt; Heimgartner, Heinz (1983). Photochemisch induzierte Reaktionen von 3-Amino-2H-azirinen. Helvetica Chimica Acta, 66:262-295.

Stegmann, Werner; Uebelhart, Peter; Heimgartner, Heinz (1983). Spirocyclische 3-Oxazoline durch 1,3-dipolare Cycloaddition von Benzonitrilio-2-propanid mit 1,4-Chinonen. Helvetica Chimica Acta, 66:2252-2268.


Obrecht, Daniel; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz (1982). 1,3-Dipolare Cycloadditionen von 2-(Benzonitrilio)-2-propanid mit 4,4-Dimethyl-2-phenyl-2-thiazolin-5-thion und Schwefelkohlenstoff. Helvetica Chimica Acta, 65:1825-1836.

Jenny, Christjohannes; Obrecht, Daniel; Heimgartner, Heinz (1982). Additionsreaktionen von 2-Thiazolin-5-thionen mit Acetylenen. Helvetica Chimica Acta, 65(8):2583-2586.

Dähler, Marlise; Prewo, Roland; Bieri, Jost H; Heimgartner, Heinz (1982). Reaktion von 3-Dimethylamino-2,2-dimethyl-2H-azirin mit 6-Methyluracil; Kristallstruktur der Reaktionsprodukte. Helvetica Chimica Acta, 65:2302-2312.

Inada, Akira; Heimgartner, Heinz (1982). Übergangsmetall-katalysierte Additionsreaktionen von 3-Phenyl-2H-azirinen und Acetylencarbonsäureestern. Helvetica Chimica Acta, 65(5):1489-1498.


Prewo, Roland; Bieri, Jost H; Widmer, Ulrich; Heimgartner, Heinz (1981). Kristallstruktur eines Tetrahydro-1(1H)-isoindolons. Helvetica Chimica Acta, 64(5):1515-1521.

Link, Helmut; Bernauer, Karl; Daly, John J; Chaloupka, Stanislav; Heimgartner, Heinz (1981). Reaktion von 3-Dimethylamino-2,2-dimethyl-2H-azirin mit Barbitursäure. Helvetica Chimica Acta, 64(1):49-63.

Obrecht, Daniel; Heimgartner, Heinz (1981). Selektive Umfunktionalisierung der terminalen Amidgruppe offenkettiger Polyamide via 2-Oxazolin-5-one als Zwischenstufen. Helvetica Chimica Acta, 64(2):482-487.


Chaloupka, Stanislav; Bieri, Jost H; Heimgartner, Heinz (1980). Struktur des Hydrazinolyseproduktes von N-(3-Oxo-1-isoindolinyliden)alanin-äthylester. Helvetica Chimica Acta, 63(7):1797-1804.


Schmid, Ursula; Heimgartner, Heinz; Schmid, Hans (1979). Additionsreaktion von 3-Dimethylamino-2,2-dimethyl-2H-azirin mit Phenylisothiocyanat. Helvetica Chimica Acta, 62(1):160-170.

Mukherjee-Müller, Gabriele; Heimgartner, Heinz; Schmid, Hans (1979). Additionsreaktionen von 3-Dimethylamino-2,2-dimethyl-2H-azirin an Phenylisocyanat und Diphenylketen. Helvetica Chimica Acta, 62(5):1429-1441.

Bruhn, Jens; Heimgartner, Heinz; Schmid, Hans (1979). Die Cope-Umlagerung als Prinzip einer repetierbaren Ringerweiterung. Helvetica Chimica Acta, 62(8):2630-2654.

Inada, Akira; Heimgartner, Heinz; Schmid, Hans (1979). Molybdenum hexacarbonyl-induced reactions of 3-aryl-2h-azirines and acetylenes. Tetrahedron Letters, (32):2983-2986.

Chaloupka, Stanislav; Heimgartner, Heinz (1979). Reaktion von 3-Amino-2H-azirinen mit Diphenylcyclopropenthion. Helvetica Chimica Acta, 62(1):86-89.

Mukherjee-Müller, Gabriele; Chaloupka, Stanislav; Heimgartner, Heinz; Schmid, Hans; Link, Helmut; Bernauer, Karl; Schönholzer, Peter; Daly, John J (1979). Reaktionen von 3-Dimethylamino-2,2-dimethyl-2H-azirin mit NH-aciden Heterocyclen; Synthese von 4H-Imidazolen. Helvetica Chimica Acta, 62(3):768-778.


Scholl, Bernhard; Bieri, Jost H; Heimgartner, Heinz (1978). 1,5,6,7-Tetrahydro-2H-[1,4]diazepin-5,7-dione aus Malonimiden und 3-Dimethylamino-2,2-dimethyl-2H-azirin. Helvetica Chimica Acta, 61(8):3050-3067.

Bieri, Jost H; Meier, Hansruedi; Heimgartner, Heinz (1978). Kristallstruktur eines überbrückten 1,2,3-Oxadiazolidin-5-ons. Helvetica Chimica Acta, 61(3):1091-1096.

Link, Helmut; Bernauer, Karl; Chaloupka, Stanislav; Heimgartner, Heinz; Schmid, Hans (1978). Reaktionsprodukte aus 3-Dimethylamino-2,2-dimethyl-2H-azirin und Phthalohydrazid bzw. Maleohydrazid. Helvetica Chimica Acta, 61(6):2116-2129.

Nakamura, Yushin; Bachmann, Kurt; Heimgartner, Heinz; Schmid, Hans; Daly, John J (1978). Stickstoffhaltige Dieisen-hexacarbonyl-Komplexe aus 3-Phenyl-2H-azirinen. Helvetica Chimica Acta, 61:589-606.

Stegmann, Werner; Uebelhart, Peter; Heimgartner, Heinz; Schmid, Hans (1978). Synthese optisch aktiver 3-phenyl-2h-azirine. Tetrahedron Letters, (34):3091-3092.

Widmer, Ulrich; Heimgartner, Heinz; Schmid, Hans (1978). Synthese von 3-Dimethylamino-3a,4,5,7a-tetrahydro-1H-isoindol-1-onen durch intramolekulare Diels-Alder-Reaktion. Helvetica Chimica Acta, 61:815-821.

Märky, Michael; Meier, Hansruedi; Wunderli, Alfred; Heimgartner, Heinz; Schmid, Hans; Hansen, Hans-Jürgen (1978). Zum photochemischen Verhalten von Sydnonen und 1,3,4-Oxadiazolin-2-onen. Helvetica Chimica Acta, 61(4):1477-1510.

Waespe, Hans-Rudolf; Heimgartner, Heinz; Schmid, Hans; Hansen, Hans-Jürgen; Paul, Henning; Fischer, Hanns (1978). Zur Photochemie von Allylaryläthern. Helvetica Chimica Acta, 61:401-429.


Lukac, Josef; Bieri, Jost H; Heimgartner, Heinz (1977). Die Struktur des Adduktes aus 3-Dimethylamino-2,2-dimethyl-2H-azirin und 3-Methyl-2,4-diphenyl-1,3-oxazolium-5-olat. Helvetica Chimica Acta, 60(5):1657-1664.

Chandrasekhar, B Parthasarathi; Heimgartner, Heinz; Schmid, Hans (1977). Reaktionen von 3-Dimethylamino-2,2-dimethyl-2H-azirin mit Phenolen und Halogenaromaten. Helvetica Chimica Acta, 60(227):2270-2287.

Chaloupka, Stanislav; Vittorelli, Piero; Heimgartner, Heinz; Schmid, Hans; Bernauer, Karl; Link, Helmut; Oberhänsli, Willi E (1977). Synthese und Reaktionen 8-gliedriger Heterocyclen aus 3-Dimethylamino-2,2-dimethyl-2H-azirin und Saccharin bzw. Phthalimid. Helvetica Chimica Acta, 60(7):2476-2495.

Meier, Hansruedi; Heimgartner, Heinz (1977). Thermisch und photochemisch induzierte intramolekulare, 1,3-dipolare Cycloadditionen von 5-(2-Allyloxyphenyl)-2-phenyltetrazol. Helvetica Chimica Acta, 60(297):3035-3038.

Wehrli, Rudolf; Heimgartner, Heinz; Schmid, Hans; Hansen, Hans-Jürgen (1977). Thermische (E),(Z)-Isomerisierungen bei substituierten Propenylbenzolen. Helvetica Chimica Acta, 60(6):2034-2061.

Meier, Hansruedi; Heimgartner, Heinz; Schmid, Hans (1977). Thermische und photochemisch induzierte intramolekulare, 1,3-dipolare Cycloadditionen von 4-Phenyl-3-(2-allylphenyl)-sydnon. Helvetica Chimica Acta, 60(3):1087-1090.

Gerber, Ulrich; Heimgartner, Heinz; Schmid, Hans; Heinzelmann, Willy (1977). Zur Regioselektivitat von Cycloadditionen photochemisch erzeugter Benzonitril-isopropylide. Helvetica Chimica Acta, 60(3):687-696.


Schmid, Ursula; Heimgartner, Heinz; Schmid, Hans; Oberhänsli, Willi E (1976). Additionsreaktionen von 3-Dimethylamino-2,2-dimethyl-2H-azirin an Isothiocyanate. Helvetica Chimica Acta, 59(8):2768-2785.

Chaloupka, Stanislav; Heimgartner, Heinz; Schmid, Hans; Link, Helmut; Schönholzer, Peter; Bernauer, Karl (1976). Herstellung und Reaktionen der valenzpolaromeren Verbindung (4,4-Dimethyl-2-thiazolin-5-dimethyliminium)-2-thiolat - (1-Dimethylthiocarbamoyl-1-methyl-äthyl)-isothiocyanat aus 3-Dimethylamino-2,2-dimethyl-2H-azirin und Schwefelkohlenstoff. Helvetica Chimica Acta, 59(7):2566-2591.

Dietliker, Kurt; Gilgen, Paul; Heimgartner, Heinz; Schmid, Hans (1976). Photochemie von in 4-Stellung substituierten 5-Methyl-3-phenyl-isoxazole. Helvetica Chimica Acta, 59(6):2074-2099.

Gakis, Nikolas; Märky, Michael; Hansen, Hans-Jürgen; Heimgartner, Heinz; Schmid, Hans; Oberhänsli, Willi E (1976). Photochemische Synthese von 4-Phenyl-3-oxazolin-5-onen und deren thermische Dimerisierung. Helvetica Chimica Acta, 59(6):2149-2167.

Stegmann, Werner; Gilgen, Paul; Heimgartner, Heinz; Schmid, Hans (1976). Photoinduzierte Cycloadditionen von 2,2-Dimethyl-3-phenyl-2H-azirin an Nitrile und "push-pull"-Olefine. Helvetica Chimica Acta, 59(4):1018-1027.


Chandrasekhar, B Parthasarathi; Schmid, Ursula; Schmid, Rudolf; Heimgartner, Heinz; Schmid, Hans (1975). Additionen von 2,2-Dimethyl-3-dimethylamino-2H-azirin an 2-Formyl-cycloalkanone und Sulfinsäuren. Helvetica Chimica Acta, 58(4):1191-1200.

Schmid, Ursula; Heimgartner, Heinz; Schmid, Hans; Schönholzer, Peter; Link, Helmut; Bernauer, Karl (1975). Die Struktur einer stabilen dipolaren Verbindung aus 2,2-Dimethyl-3-dimethylamino-2H-azirin und Benzoylisothiocyanat. Helvetica Chimica Acta, 58(7):2222-2227.

Widmer, Ulrich; Heimgartner, Heinz; Schmid, Hans (1975). Photochemie von 1,1-Dimethyl-4-phenyl- und 1-Methyl-1-phenyl-1,2-dihydronaphthalin; Nachweis einer photochemischen, sigmatropischen [1,7]H-Verschiebung. Helvetica Chimica Acta, 58(7):2210-2222.

Gakis, Nikolas; Heimgartner, Heinz; Schmid, Hans (1975). Photochemische Cycloadditionen von 3-Phenyl-2H-azirinen mit Benzoyl-, Äthoxycarbonyl- und Vinylphosphonaten. Helvetica Chimica Acta, 58(3):748-760.

Orahovats, Alexander; Heimgartner, Heinz; Schmid, Hans; Heinzelmann, Willy (1975). Photochemische Erzeugung und Reaktionen des Benzonitril-benzylids. Helvetica Chimica Acta, 58(8):2662-2677.

Gilgen, Paul; Hansen, Hans-Jürgen; Heimgartner, Heinz; Sieber, Willi; Uebelhart, Peter; Schmid, Hans; Schönholzer, Peter; Oberhänsli, Willi E (1975). Photoinduzierte Reaktionen von 3-Phenyl-2H-azirinen mit Carbonsäureestern. Helvetica Chimica Acta, 58(6):1739-1768.


Vittorelli, Piero; Heimgartner, Heinz; Schmid, Hans; Hoet, P; Ghosez, Leon (1974). Addition of carboxylic acidis and cyclic 1,3-diketones to 2-dimethylamino-3,3-dimethyl-1-azirine. Tetrahedron, 30:3737-3740.

Schmid, Ursula; Gilgen, Paul; Heimgartner, Heinz; Hansen, Hans-Jürgen; Schmid, Hans (1974). Photochemische Cycloadditionen von 3-Phenyl-2H-azirinen an Carbonsäurechloride. Helvetica Chimica Acta, 57(5):1393-1403.

Claus, Peter; Gilgen, Paul; Hansen, Hans-Jürgen; Heimgartner, Heinz; Jackson, Barry; Schmid, Hans (1974). Photochemische Cycloadditionen von 3-Phenyl-2H-azirinen mit Ketonen, Acylcyaniden und Ketoestern. Helvetica Chimica Acta, 57(7):2173-2192.

Gakis, Nikolas; Heimgartner, Heinz; Schmid, Hans (1974). Photochemische Cycloadditionen von 3-Phenyl-2H-azirinen mit Triphenyl-vinylphosphoniumbromid. Helvetica Chimica Acta, 57(5):1403-1407.

Gilgen, Paul; Heimgartner, Heinz; Schmid, Hans (1974). Photoinduzierte 1,3-dipolare Cycloaddition von 3-Phenyl-2H-azirinen an Azodicarbonsäure-diäthylester. Helvetica Chimica Acta, 57(5):1382-1392.

Orahovats, Alexander; Heimgartner, Heinz; Schmid, Hans; Heinzelmann, Willy (1974). Photoinduzierte Cycloadditionen von aliphatischen 2H-Azirinen. Helvetica Chimica Acta, 57(8):2626-2633.

Gilgen, Paul; Jackson, Barry; Hansen, Hans-Jürgen; Heimgartner, Heinz; Schmid, Hans (1974). Synthese von 2H-Isoindol-4,7-dionen durch photochemische Cycloaddition von 2,3-Diphenyl-2H-azirin an 1,4-Chinone. Helvetica Chimica Acta, 57(8):2634-2643.


Heimgartner, Heinz; Zsindely, Janos; Hansen, Hans-Jürgen; Schmid, Hans (1973). Aromatische [1,5s]-sigmatropische H-Verschiebungen in Arylallenen. Helvetica Chimica Acta, 56(8):2924-2945.

Giezendanner, Heinz; Heimgartner, Heinz; Jackson, Barry; Winkler, Tammo; Hansen, Hans-Jürgen; Schmid, Hans (1973). Photochemische Cycloadditionen von 3-Phenyl-2H-azirinen mit Aldehyden. Helvetica Chimica Acta, 56(7):2611-2627.

Orahovats, Alexander; Jackson, Barry; Heimgartner, Heinz; Schmid, Hans (1973). Photoinduzierte Cycloadditionen von 3-Benzyl-2H-azirin. Helvetica Chimica Acta, 56(6):2007-2011.

Narasimhan, Nurani S; Heimgartner, Heinz; Hansen, Hans-Jürgen; Schmid, Hans (1973). Thermische Reaktionen mit 3-Phenyl-2H-azirinen; 1,3-dipolare Cycloadditionen und En-Reaktionen. Helvetica Chimica Acta, 56(4):1351-1370.


Heimgartner, Heinz; Zsindely, Janos; Hansen, Hans-Jürgen; Schmid, Hans (1972). Die Dienol-Benzol-Umlagerung von Propargylcyclohexadienolen: aromatische [1,2]-, [3,3]- und [3,4]-sigmatropische Umlagerungen. Helvetica Chimica Acta, 55(4):1113-1141.

Sieber, Willi; Heimgartner, Heinz; Hansen, Hans-Jürgen; Schmid, Hans (1972). Photochemisches Verhalten von 1- und 2-alkylierten 1,2-Dihydronaphthalinen bei tiefen Temperaturen. Helvetica Chimica Acta, 55(8):3005-3026.

Heimgartner, Heinz; Hansen, Hans-Jürgen; Schmid, Hans (1972). Thermisches Verhalten von 1,2-Dipropenylbenzolen. Helvetica Chimica Acta, 55(5):1385-1403.


Heimgartner, Heinz; Ulrich, Linus; Hansen, Hans-Jürgen; Schmid, Hans (1971). Photochemisches Verhalten von 1- und 2-alkylierten 1,2-Dihydronaphtalinen. Helvetica Chimica Acta, 54(7):2313-2354.


Heimgartner, Heinz; Zsindely, Janos; Hansen, Hans-Jürgen; Schmid, Hans (1970). Thermisches Verhalten von Mesitylallenen; Beispiel einer aromatischen [1,5s]-sigmatropischen H-Verschiebung. Helvetica Chimica Acta, 53(5):1212-1215.

Heimgartner, Heinz; Hansen, Hans-Jürgen; Schmid, Hans (1970). Thermisches Verhalten von o-Dipropenylbenzol, Beispiel einer aromatischen [1,7]-sigmatropischen H-Verschiebung. Helvetica Chimica Acta, 53(1):173-176.

This list was generated on Sun May 19 00:24:41 2024 CEST.